SCHEMBL5822282

SCHEMBL5822282

O=C(CCl)NCCN1CCCCC1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.58
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
CA9 Q16790 3/20 0.58
ALDH1A1 P00352 4/20 0.57
GAA P10253 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
KDM4E B2RXH2 2/20 0.54
NPC1 O15118 1/20 0.53
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.49
POLB P06746 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CNR1 P21554 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11028517 0.98 CA12 (0.56) CA12CA1CA2CA9ALDH1A1
SCHEMBL8256720 0.89 HRH3 (0.53) CA12CA1CA2CA9ALDH1A1
SCHEMBL11025226 0.87 SMN1; SMN2 (0.55) ALDH1A1SMN1; SMN2KDM4EMAPTCYP1A2
SCHEMBL11027232 0.86 SMN1; SMN2 (0.54) ALDH1A1GAASMN1; SMN2MAPTCYP1A2
SCHEMBL13661591 0.84 MAPT (0.70) CA12CA1CA2CA9ALDH1A1
SCHEMBL4283848 0.84 ALDH1A1 (0.81) CA12CA1CA2CA9ALDH1A1
SCHEMBL84849 0.82 ALDH1A1 (0.57) CA12CA1CA2CA9ALDH1A1
SCHEMBL18629170 0.82 CA12 (0.56) CA12CA1CA2CA9ALDH1A1
SCHEMBL20249046 0.82 CA12 (0.56) CA12CA1CA2CA9ALDH1A1
SCHEMBL11026192 0.82 HDAC2 (0.51) ALDH1A1GAASMN1; SMN2POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174488-A1 SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS INSILICO MEDICINE IP LIMITED (HK) 2023-06-08 US disclosed
US-20070037822-A1 Azinone and diazinone V3 inhibitors for depression and stress disorders PHARMACOPEIA DRUG DISCOVERY, INC. (US) 2007-02-15 US disclosed
US-20070037822-A1 Azinone and diazinone V3 inhibitors for depression and stress disorders PHARMACOPEIA DRUG DISCOVERY, INC. (US) 2007-02-15 US disclosed
WO-2006133242-A2 AZINONE AND DIAZINONE V3 INHIBITORS FOR DEPRESSION AND STRESS DISORDERS PHARMACOPEIA, INC. (US) 2006-12-14 WO disclosed
US-20060135553-A1 Imidazole derivatives PHENOMIX CORPORATION 2006-06-22 US disclosed
WO-2006050162-A2 IMIDAZOLE DERIVATIVES PHENOMIX CORPORATION (US) 2006-05-11 WO disclosed
EP-0040793-B1 NOVEL QUINAZOLINE-DIONE COMPOUNDS, PROCESS FOR PRODUCTION THEREOF AND PHARMACEUTICAL USE THEREOF Ishikawa, Masayuki (JP) 1985-08-28 EP disclosed
US-4405623-A HYPOTENSIVE AGENTS, VASODILATORS MASAYUKI ISHIKAWA (JP) 1983-09-20 US disclosed
EP-0040793-A1 Novel quinazoline-dione compounds, process for production thereof and pharmaceutical use thereof Ishikawa, Masayuki (JP) 1981-12-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060135553-A1 Imidazole derivatives FLT4, NOS2, FLT1 CA12 4674/4885CA1 4663/4885CA2 2855/4885
US-20070037822-A1 Azinone and diazinone V3 inhibitors for depression and stress disorders HTR3C, HTR3A, AZI2 CA12 4808/4885CA1 3982/4885CA2 4338/4885
US-20230174488-A1 SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS ACE2, SARS1, ACE CA12 2497/4885CA1 4450/4885CA2 1997/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.