SCHEMBL5845485

SCHEMBL5845485

CS(=O)(=O)O.N[C@@H](CC(=O)O)c1ccccc1

nearest known ligand 0.49

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GABBR2 O75899 1/20 0.49
GABBR1 Q9UBS5 1/20 0.49
GBA1 P04062 1/20 0.47
CYP2C19 P33261 2/20 0.45
ATM Q13315 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
SRC P12931 1/20 0.43
EEF2K O00418 1/20 0.42
TPH1 P17752 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5846637 1.00 KMT2A (0.49) KMT2ASMN1; SMN2GABBR2GABBR1GBA1
SCHEMBL5845499 1.00 KMT2A (0.49) KMT2ASMN1; SMN2GABBR2GABBR1GBA1
SCHEMBL123765 0.89 GABBR2 (0.59) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
SCHEMBL288753 0.89 GABBR2 (0.59) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
SCHEMBL59840 0.89 GABBR2 (0.59) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
Hydrochloric Acid SCHEMBL3874351 0.87 GABBR2 (0.57) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
SCHEMBL9386161 0.87 GABBR2 (0.57) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
Hydrochloric Acid SCHEMBL2934796 0.87 GABBR2 (0.57) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
Hydrochloric Acid SCHEMBL4150999 0.87 GABBR2 (0.57) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19
Acetamide SCHEMBL27677566 0.85 GABBR2 (0.52) KMT2ASMN1; SMN2GABBR2GABBR1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7015348-B2 Method for producing an optically active β-amino acid TAKASAGO INTERNATIONAL CORPORATION (JP) 2006-03-21 US claimed
EP-1386901-B1 Method for producing an optically active beta-amino acid TAKASAGO PERFUMERY CO LTD (JP) 2015-07-01 EP disclosed
US-20060122418-A1 Method for producing an optically active beta-amino acid MATSUMURA KAZUHIKO 2006-06-08 US disclosed
US-7015348-B2 Method for producing an optically active β-amino acid TAKASAGO INTERNATIONAL CORPORATION (JP) 2006-03-21 US disclosed
US-20040023344-A1 Method for producing an optically activ beta-amino acid TAKASAGO INTERNATIONAL CORPORATION (JP) 2004-02-05 US disclosed
EP-1386901-A1 Method for producing an optically active beta-amino acid Takasago International Corporation (JP) 2004-02-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060122418-A1 Method for producing an optically active beta-amino acid AADAT, DAO, BCAT2 KMT2A 2862/4885SMN1; SMN2 3286/4885GABBR2 907/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.