SCHEMBL5867337

SCHEMBL5867337

CCn1nc(C)cc1C1CCN(CCC(NS(=O)(=O)c2ccc(Br)cc2)c2ccccc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
PRCP P42785 2/20 0.39
HTR1A P08908 3/20 0.39
HTR7 P34969 3/20 0.39
CCR5 P51681 9/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5448681 0.99 KMT2A (0.41) KMT2APRCPHTR1AHTR7CCR5
SCHEMBL5467769 0.94 CCR5 (0.42) KMT2APRCPCCR5ALDH1A1
SCHEMBL5452648 0.94 CCR5 (0.42) KMT2APRCPCCR5ALDH1A1
SCHEMBL5868117 0.92 HTR7 (0.42) KMT2APRCPHTR1AHTR7CCR5
SCHEMBL5867355 0.92 SIGMAR1 (0.43) KMT2APRCPHTR1AHTR7CCR5
Hydrochloric Acid SCHEMBL5459369 0.91 HTR7 (0.41) KMT2APRCPHTR1AHTR7CCR5
Hydrochloric Acid SCHEMBL5463380 0.91 SIGMAR1 (0.43) KMT2APRCPHTR1AHTR7CCR5
SCHEMBL6715399 0.86 PRCP (0.40) KMT2APRCPCCR5
Hydrochloric Acid SCHEMBL5867442 0.85 TP53 (0.43) KMT2APRCPCCR5ALDH1A1HTT
SCHEMBL5458123 0.84 KMT2A (0.44) KMT2AHTR1AHTR7CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7153868-B2 N-(3-(4-substituted-1-piperidinyl)-1-phenylpropyl) substituted sulfonamides as NK-3 receptor antagonists MERCK SHARP & DOHME LTD. 2006-12-26 US claimed