SCHEMBL5867355

SCHEMBL5867355

CCn1nc(C)cc1C1CCN(CCC(NS(=O)(=O)c2ccc(F)cc2)c2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
CCR5 P51681 14/20 0.42
KMT2A Q03164 1/20 0.41
HTR7 P34969 3/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR1A P08908 2/20 0.39
PRCP P42785 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5463380 0.99 SIGMAR1 (0.43) SIGMAR1CCR5KMT2AHTR7HTR2A
SCHEMBL5467769 0.94 CCR5 (0.42) CCR5KMT2APRCP
SCHEMBL5452648 0.94 CCR5 (0.42) CCR5KMT2APRCP
SCHEMBL5867337 0.92 KMT2A (0.41) CCR5KMT2AHTR7HTR1APRCP
Hydrochloric Acid SCHEMBL5448681 0.91 KMT2A (0.41) CCR5KMT2AHTR7HTR1APRCP
SCHEMBL5868117 0.87 HTR7 (0.42) CCR5KMT2AHTR7HTR1APRCP
SCHEMBL6715399 0.86 PRCP (0.40) CCR5KMT2APRCP
Hydrochloric Acid SCHEMBL5459369 0.86 HTR7 (0.41) CCR5KMT2AHTR7HTR1APRCP
SCHEMBL5458123 0.84 KMT2A (0.44) CCR5KMT2AHTR7HTR1A
Hydrochloric Acid SCHEMBL5458549 0.83 KMT2A (0.43) CCR5KMT2AHTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7153868-B2 N-(3-(4-substituted-1-piperidinyl)-1-phenylpropyl) substituted sulfonamides as NK-3 receptor antagonists MERCK SHARP & DOHME LTD. 2006-12-26 US claimed