SCHEMBL5869919

SCHEMBL5869919

CC(C)CC(NC(Cc1ccc(NC(=O)c2ccncc2)cn1)C(=O)O)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 2/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
HTT P42858 1/20 0.41
AKT1 P31749 1/20 0.40
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
PGGT1B P53609 1/20 0.39
DGAT1 O75907 1/20 0.39
NPC1 O15118 1/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
JAK2 O60674 1/20 0.39
TYK2 P29597 1/20 0.39
ACE2 Q9BYF1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8255230 1.00 KMT2A (0.47) KMT2ARAB9AKDM4EGAAALDH1A1
SCHEMBL8256279 0.85 RAB9A (0.42) RAB9AKDM4EALDH1A1NPC1ACE2
SCHEMBL5869809 0.85 RAB9A (0.42) RAB9AKDM4EALDH1A1NPC1ACE2
SCHEMBL8249899 0.81 ALDH1A1 (0.56) KMT2ARAB9AALDH1A1TP53HTT
SCHEMBL5869783 0.81 ALDH1A1 (0.56) KMT2ARAB9AALDH1A1TP53HTT
SCHEMBL5869254 0.77 TAS1R3 (0.50) DGAT1
SCHEMBL8256132 0.77 TAS1R3 (0.50) DGAT1
SCHEMBL8254618 0.73 PTPRA (0.54) ALDH1A1MAPK1FNTAFNTBPGGT1B
SCHEMBL5870034 0.73 PTPRA (0.54) ALDH1A1MAPK1FNTAFNTBPGGT1B
SCHEMBL23303692 0.72 CA2 (0.62) KMT2AKDM4EALDH1A1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7045532-B2 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-05-16 US disclosed
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. 2004-04-29 US disclosed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040082496-A1 ACE-2 modulating compounds and methods of use thereof ACE, ACE2, AGTR2 KMT2A 1880/4885RAB9A 2897/4885KDM4E 2662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.