SCHEMBL5885151

SCHEMBL5885151

CON(C(N)=O)C(=O)C(O)[CH]Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LAP3 P28838 1/20 0.35
ALOX5 P09917 4/20 0.35
SLC15A1 P46059 1/20 0.35
HTT P42858 1/20 0.34
EPHX1 P07099 2/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
FAAH O00519 1/20 0.33
ABCB1 P08183 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
SRR Q9GZT4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6052877 1.00 LAP3 (0.35) LAP3ALOX5SLC15A1HTTEPHX1
SCHEMBL6342303 1.00 LAP3 (0.35) LAP3ALOX5SLC15A1HTTEPHX1
SCHEMBL3131488 0.81 HPGD (0.38) ALOX5SLC15A1EPHX1HPGD
SCHEMBL8411597 0.81 FAAH (0.41) LAP3FAAHABCB1HPGDTSHR
SCHEMBL6342050 0.80 ALOX5 (0.36) LAP3ALOX5SLC15A1EPHX1
SCHEMBL6164405 0.78 LAP3 (0.36) LAP3ALOX5L3MBTL1
SCHEMBL8411083 0.77 MMP9 (0.43) HPGD
SCHEMBL6354283 0.76 UBE2N (0.36) HPGDTSHR
SCHEMBL28026869 0.75 EPHX1 (0.46) SLC15A1EPHX1L3MBTL1SRR
SCHEMBL27660866 0.75 EPHX1 (0.46) SLC15A1EPHX1L3MBTL1SRR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6992101-B2 N-(indole-2-carbonyl) and H-thieno[2,3-b]pyrrole-5-carboxamide anti-diabetic agents PFIZER, INC. (US) 2006-01-31 US disclosed
EP-1562899-A2 N-(INDOLE-2-CARBONYL)AMIDES AS ANTI-DIABETIC AGENTS Pfizer Products Inc. (US) 2005-08-17 EP disclosed
US-20040157907-A1 Anti-diabetic agents PFIZER INC 2004-08-12 US disclosed
WO-2004041780-A2 N-(INDOLE-2-CARBONYL) AMIDES AS ANTI-DIABETIC AGENTS PFIZER PRODUCTS INC. (US) 2004-05-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157907-A1 Anti-diabetic agents GPR119, INSR, IRS1 LAP3 2259/4885ALOX5 933/4885SLC15A1 715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.