SCHEMBL5887436

SCHEMBL5887436

Cc1ccc(C2=C(Cl)C(Cl)=C(c3ccccc3Cl)[CH]C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.36
KMT2A Q03164 5/20 0.35
POLB P06746 1/20 0.35
HSD11B1 P28845 3/20 0.34
MEN1 O00255 4/20 0.34
MAPT P10636 3/20 0.33
HPGD P15428 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ALOX15 P16050 2/20 0.33
ALDH1A1 P00352 2/20 0.33
USP2 O75604 1/20 0.33
TP53 P04637 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MITF O75030 1/20 0.33
HTT P42858 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047645 0.81 HSD11B1 (0.38) HSD11B1
SCHEMBL6047589 0.80 PTGS1 (0.35) KMT2AMEN1NPC1RAB9ANFKB1
SCHEMBL5887404 0.77 L3MBTL1 (0.40) KMT2AMEN1MAPTHPGDALDH1A1
SCHEMBL1045000 0.73 CYP2A6 (0.65) CYP2A6KMT2APOLBHSD11B1MEN1
SCHEMBL5887582 0.69 TSHR (0.43) KMT2APOLBMEN1MAPTHPGD
SCHEMBL5887426 0.66 MEN1 (0.34) CYP2A6KMT2APOLBMEN1HPGD
Bicarbonate SCHEMBL27450693 0.66 CYP2A6 (0.59) CYP2A6KMT2AMEN1NPC1RAB9A
SCHEMBL11260432 0.65 HSD11B1 (0.47) CYP2A6KMT2AHSD11B1MEN1MAPT
SCHEMBL1047922 0.63 CNR2 (0.50) CYP2A6
SCHEMBL6047627 0.62 CYP2A6 (0.39) CYP2A6KMT2APOLBHSD11B1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed