SCHEMBL5894508

SCHEMBL5894508

[O-][n+]1ccc2ccccc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
MAPT P10636 3/20 0.38
HPGD P15428 2/20 0.37
GLA P06280 1/20 0.37
ACHE P22303 1/20 0.37
NCF1 P14598 3/20 0.37
CYP1A2 P05177 2/20 0.37
NOS2 P35228 1/20 0.37
BACE1 P56817 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
NQO2 P16083 1/20 0.36
EGFR P00533 1/20 0.35
KDM4E B2RXH2 4/20 0.34
LMNA P02545 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
PKM P14618 1/20 0.34
ATM Q13315 1/20 0.33
MGAM O43451 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28614872 0.73 ALDH1A1 (0.39) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL5152358 0.70 ALDH1A1 (0.40) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL5894504 0.70 ALDH1A1 (0.41) ALDH1A1MAPTCYP1A2CA12CA9
SCHEMBL28921608 0.68 ALDH1A1 (0.35) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL5894552 0.68 ALDH1A1 (0.39) ALDH1A1MAPTKDM4ELMNANPC1
SCHEMBL996754 0.68 CA12 (0.41) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL18095030 0.68 MAPT (0.38) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL8821267 0.68 EGFR (0.40) ALDH1A1MAPTHPGDGLAACHE
SCHEMBL22144248 0.67 NCF1 (0.36) ALDH1A1MAPTACHENCF1CYP1A2
SCHEMBL22124480 0.66 RXFP1 (0.40) ALDH1A1MAPTHPGDCYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119638634-A Cinnoline-2-oxide compound, preparation method and application thereof 上海赛默罗生物科技有限公司 2025-03-18 CN claimed
EP-3849984-A1 1-ISOPROPYL-3-METHYL-8- (PYRIDIN-3-YL) -1, 3-DIHYDRO-2H-IMIDAZO [4, 5-C] CINNOLIN-2-ONE AS SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF Suzhou Zanrong Pharma Limited (CN) 2021-07-21 EP claimed
WO-2020052688-A1 1-ISOPROPYL-3-METHYL-8- (PYRIDIN-3-YL) -1, 3-DIHYDRO-2H-IMIDAZO [4, 5-c] CINNOLIN-2-ONE AS SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2020-03-19 WO claimed
WO-2019057757-A1 1,3-DIHYDROIMIDAZO[4,5-C]CINNOLIN-2-ONE COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2019-03-28 WO claimed
US-20060156485-A1 Keratin dyeing compounds, keratin dyeing compositions containing them, and use thereof THE PROCTER & GAMBLE COMPANY (US) 2006-07-20 US claimed
CN-119638634-B Cinnoline-2-oxide compound, preparation method and application thereof 上海赛默罗生物科技有限公司 2026-01-30 CN disclosed
CN-119638634-B Cinnoline-2-oxide compound, preparation method and application thereof 上海赛默罗生物科技有限公司 2026-01-30 CN disclosed
CN-119638634-A Cinnoline-2-oxide compound, preparation method and application thereof 上海赛默罗生物科技有限公司 2025-03-18 CN disclosed
CN-119638634-A Cinnoline-2-oxide compound, preparation method and application thereof 上海赛默罗生物科技有限公司 2025-03-18 CN disclosed
CN-119638634-A Cinnoline-2-oxide compound, preparation method and application thereof 上海赛默罗生物科技有限公司 2025-03-18 CN disclosed
US-20240207263-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2024-06-27 US disclosed
EP-4308569-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF Suzhou Zanrong Pharma Limited (CN) 2024-01-24 EP disclosed
EP-3849984-A1 1-ISOPROPYL-3-METHYL-8- (PYRIDIN-3-YL) -1, 3-DIHYDRO-2H-IMIDAZO [4, 5-C] CINNOLIN-2-ONE AS SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF Suzhou Zanrong Pharma Limited (CN) 2021-07-21 EP disclosed
CN-112752758-A 1-isopropyl-3-methyl-8- (pyridin-3-yl) -1, 3-dihydro-2H-imidazo [4,5-c ] cinnolin-2-one as selective modulator of ataxia-telangiectasia mutated (ATM) kinase and uses thereof 苏州赞荣医药科技有限公司 2021-05-04 CN disclosed
CN-111344293-A 1, 3-dihydroimidazo [4, 5-c ] cinnolin-2-one compounds and their use in the treatment of cancer 阿斯利康(瑞典)有限公司 2020-06-26 CN disclosed
CN-111344293-A 1, 3-dihydroimidazo [4, 5-c ] cinnolin-2-one compounds and their use in the treatment of cancer 阿斯利康(瑞典)有限公司 2020-06-26 CN disclosed
WO-2020052688-A1 1-ISOPROPYL-3-METHYL-8- (PYRIDIN-3-YL) -1, 3-DIHYDRO-2H-IMIDAZO [4, 5-c] CINNOLIN-2-ONE AS SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2020-03-19 WO disclosed
WO-2020052688-A1 1-ISOPROPYL-3-METHYL-8- (PYRIDIN-3-YL) -1, 3-DIHYDRO-2H-IMIDAZO [4, 5-c] CINNOLIN-2-ONE AS SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2020-03-19 WO disclosed
WO-2019057757-A1 1,3-DIHYDROIMIDAZO[4,5-C]CINNOLIN-2-ONE COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2019-03-28 WO disclosed
US-20060156485-A1 Keratin dyeing compounds, keratin dyeing compositions containing them, and use thereof THE PROCTER & GAMBLE COMPANY (US) 2006-07-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060156485-A1 Keratin dyeing compounds, keratin dyeing compositions containing them, and use thereof KRT18, TUBB6, DNMT1 ALDH1A1 385/4885MAPT 1322/4885HPGD 158/4885
US-20240207263-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF ATM, CHEK2, CHEK1 ALDH1A1 3923/4885MAPT 1185/4885HPGD 3123/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.