SCHEMBL5907151

SCHEMBL5907151

Nc1nc(=O)cc(Cc2ccccc2)[nH]1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.56
XDH P47989 3/20 0.52
LTB4R Q15722 1/20 0.51
PARP1 P09874 1/20 0.50
PNP P00491 4/20 0.49
BACE1 P56817 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ADORA1 P30542 1/20 0.47
HCAR2 Q8TDS4 1/20 0.44
DAO P14920 1/20 0.44
DHFR P00374 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21332729 0.77 PARP1 (0.50) AOC3XDHLTB4RPARP1PNP
SCHEMBL9878574 0.76 POLB (0.61) XDHPARP1SMN1; SMN2ADORA1HCAR2
SCHEMBL5907152 0.73 BACE1 (0.74) XDHLTB4RPNPBACE1
SCHEMBL3723702 0.73 BACE1 (0.44) XDHPARP1PNPBACE1ADORA1
SCHEMBL12598581 0.72 AOC3 (1.00) AOC3XDHLTB4RPARP1PNP
SCHEMBL10843644 0.70 XDH (0.54) XDHPARP1ADORA1
SCHEMBL9879243 0.70 BACE1 (0.54) XDHBACE1SMN1; SMN2ADORA1HCAR2
SCHEMBL9879095 0.70 MEN1 (0.54) SMN1; SMN2ADORA1DAO
SCHEMBL12956835 0.70 PNP (0.62) XDHLTB4RPNPSMN1; SMN2DHFR
SCHEMBL7106470 0.69 PARP1 (0.65) PARP1SMN1; SMN2ADORA1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114716961-B Self-complementary quadruple hydrogen bond supermolecule hot melt adhesive and synthesis method thereof 郑州大学 2023-06-23 CN disclosed
CN-114716961-A Self-complementary quadruple hydrogen bond supramolecular hot melt adhesive and synthesis method thereof 郑州大学 2022-07-08 CN disclosed
US-20060106044-A1 Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4-oxopyrimidines IDENIX PHARMACEUTICALS INC. (US) 2006-05-18 US disclosed
US-20040092539-A1 Substituted 6-benzyl-4-oxopyrimidines, process for their preparation and pharmaceutical compositions containing them COLLA PAOLO LA (IT) 2004-05-13 US disclosed
US-20030225114-A1 Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4- oxopyrimidines IDENIX PHARMACEUTICALS, INC. 2003-12-04 US disclosed
US-6635636-B1 Reverse transcriptase inhibitors; human immunodeficiency virus and acquired immune deficiency syndrome IDENIX PHARMACEUTICALS, INC. 2003-10-21 US disclosed
US-6545007-B2 Topically applying to the skin or epithelial tissue of a human an effective amount of a dihydro-alkyloxy-benzyl-oxopyrimidine compound for inhibiting sexual transmission of HIV IDENIX (CAYMAN) LIMITED (KY) 2003-04-08 US disclosed
US-20030008887-A1 Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4-oxopyrimidines IDENIX PHARMACEUTICALS INC. 2003-01-09 US disclosed
EP-1098887-A1 SUBSTITUTED 6-BENZYL-4-OXOPYRIMIDINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Novirio Pharmaceuticals Limited (KY) 2001-05-16 EP disclosed
WO-2000003998-A1 SUBSTITUTED 6-BENZYL-4-OXOPYRIMIDINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NOVIRIO PHARMACEUTICALS LIMITED (KY) 2000-01-27 WO disclosed
WO-1991018887-A1 DIAMINOPYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1991-12-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106044-A1 Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4-oxopyrimidines DUT, UNG, NUDT1 AOC3 571/4885XDH 240/4885LTB4R 3107/4885
US-20030008887-A1 Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4-oxopyrimidines DUT, UNG, NUDT1 AOC3 499/4885XDH 258/4885LTB4R 2820/4885
US-20040092539-A1 Substituted 6-benzyl-4-oxopyrimidines, process for their preparation and pharmaceutical compositions containing them TYMP, UMPS, TYMS AOC3 1537/4885XDH 48/4885LTB4R 2628/4885
US-20030225114-A1 Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4- oxopyrimidines DUT, UNG, NUDT1 AOC3 499/4885XDH 258/4885LTB4R 2820/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.