SCHEMBL59342

SCHEMBL59342

CCCCCCCC=CCC=CCCCCCCCC

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.70
ALDH1A1 P00352 4/20 0.65
KDM4E B2RXH2 3/20 0.65
F7 P08709 3/20 0.65
F3 P13726 3/20 0.65
PPARG P37231 3/20 0.65
PPARD Q03181 2/20 0.65
PPARA Q07869 2/20 0.65
FABP3 P05413 2/20 0.65
DUSP3 P51452 1/20 0.65
PTPN7 P35236 1/20 0.65
FFAR1 O14842 1/20 0.65
LMNA P02545 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP19A1 P11511 1/20 0.65
FABP4 P15090 1/20 0.65
HPGD P15428 1/20 0.65
ALOX15 P16050 1/20 0.65
TSHR P16473 1/20 0.65
PTGS1 P23219 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6477506 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL6472470 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL4750573 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL6473134 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL220462 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL20503612 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL24283496 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL6476959 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL6477509 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3
SCHEMBL18035471 1.00 TRPV1 (0.70) TRPV1ALDH1A1KDM4EF7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 619 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11999754-B2 Ruthenium complexes and their use in olefin metathesis reactions APEIRON SYNTHESIS S.A. (PL) 2024-06-04 US disclosed
US-20240158439-A1 INHIBITORS OF ANTIGEN PRESENTATION BY MHC CLASS II HLA-DRB1*15:01 MOLECULES WITH ENHANCED METABOLIC STABILITY PROVID PHARMACEUTICALS INC. 2024-05-16 US disclosed
US-11976085-B2 Process for producing ruthenium complexes and intermediates thereof and their use in olefin metathesis Aperion Synthesis S.A. (PL) 2024-05-07 US disclosed
US-20240136527-A1 Binder for Secondary Battery, Negative Electrode for Secondary Battery Including the Same, and Lithium Secondary Battery Including the Same SK INNOVATION CO., LTD. (KR) 2024-04-25 US disclosed
EP-4354555-A1 BINDER FOR SECONDARY BATTERY, NEGATIVE ELECTRODE FOR SECONDARY BATTERY INCLUDING THE SAME, AND LITHIUM SECONDARY BATTERY INCLUDING THE SAME SK Innovation Co., Ltd. (KR) 2024-04-17 EP disclosed
WO-2024069256-A1 TRANSITION METAL COMPOUND, CATALYST COMPOSITION COMPRISING THE SAME, AND METHOD FOR PREPARING OLEFIN POLYMER USING THE SAME SABIC SK NEXLENE COMPANY PTE. LTD. (SG) 2024-04-04 WO disclosed
WO-2024052871-A1 NOVEL RUTHENIUM COMPLEXES, METHOD OF THEIR SYNTHESIS, INTERMEDIATE COMPOUNDS USED IN THIS METHOD, METHOD OF THEIR SYNTHESIS AND USE OF NOVEL RUTHENIUM COMPLEXES IN OLEFIN METATHESIS REACTIONS UNIWERSYTET WARSZAWSKI (PL) 2024-03-14 WO disclosed
US-20240076308-A1 PROCESS FOR PRODUCING RUTHENIUM COMPLEXES AND INTERMEDIATES THEREOF AND THEIR USE IN OLEFIN METATHESIS APEIRON SYNTHESIS SA (PL) 2024-03-07 US disclosed
EP-4112053-B1 TREATMENT OF SYNUCLEINOPATHIES DEUTSCHES ZENTRUM FUER NEURODEGENERATIVE ERKRANKUNGEN E V DZNE (DE) 2024-02-14 EP disclosed
EP-4308585-A1 INHIBITORS OF ANTIGEN PRESENTATION BY MHC CLASS II HLA-DRB1*15:01 MOLECULES WITH ENHANCED METABOLIC STABILITY Provid Pharmaceuticals Inc. (US) 2024-01-24 EP disclosed
WO-2004009610-A2 USE OF NUCLEOSIDE COMPOUNDS FOR NONSENSE SUPPRESSION AND THE TREATMENT OF GENETIC DISEASES PTC THERAPEUTICS, INC. (US) 2004-01-29 WO disclosed
WO-2004009609-A2 NUCLEOSIDE COMPOUNDS AND THEIR USE FOR TREATING CANCER AND DISEASES ASSOCIATED WITH SOMATIC MUTATIONS PTC THERAPEUTICS, INC. (US) 2004-01-29 WO disclosed
WO-2004009533-A1 ACETYLAMINO BENZOIC ACID COMPOUNDS AND THEIR USE FOR NONSENSE SUPPRESSION AND THE TREATMENT OF DISEASE PTC THERAPEUTICS, INC. (US) 2004-01-29 WO disclosed
WO-2004009563-A1 5-ARYLTETRAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND USES THEREFOR INOTEK PHARMACEUTICALS CORPORATION (US) 2004-01-29 WO disclosed
WO-2004004774-A2 COMPOSITIONS COMPRISING PANTHETINE FOR THE TREATMENT OF DYSLIPIDEMIA ESPERION THERAPEUTICS, INC. (US) 2004-01-15 WO disclosed
WO-2003105774-A2 COMPOUNDS USEFUL FOR THE TREATMENT OF CANCER, COMPOSITIONS THEREOF AND METHODS THEREWITH SIGNAL PHARMACEUTICALS, INC. (US) 2003-12-24 WO disclosed
WO-2003102151-A2 MODULATING CELL DIFFERENTIATION AND TREATING MYELOPROLIFERTIVE DISORDERS WITH JNK/MKK INHIBITORS CELGENE CORPORATION (US) 2003-12-11 WO disclosed
WO-2003099221-A2 METHODS FOR USING JNK INHIBITORS FOR TREATING OR PREVENTING DISEASE-RELATED WASTING SIGNAL PHARMACEUTICALS, INC. (US) 2003-12-04 WO disclosed
WO-2003093236-A1 1-(PYRID-2-YL)-PIPERAZINE COMPOUNDS AS METABOTROPIC GLUTAMATE RECEPTOR INHIBITOR EURO-CELTIQUE, S.A. (LU) 2003-11-13 WO disclosed
WO-2003075917-A1 COMBINATION THERAPY FOR TREATING, PREVENTING OR MANAGING PROLIFERATIVE DISORDERS AND CANCERS SIGNAL PHARMACEUTICALS, INC. (US) 2003-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240158439-A1 INHIBITORS OF ANTIGEN PRESENTATION BY MHC CLASS II HLA-DRB1*15:01 MOLECULES WITH ENHANCED METABOLIC STABILITY HLA-DRB1, HLA-B, HLA-C TRPV1 1768/4885ALDH1A1 1812/4885KDM4E 3390/4885
US-11976085-B2 Process for producing ruthenium complexes and intermediates thereof and their use in olefin metathesis POR, CYP1B1, CYP4F11 TRPV1 3244/4885ALDH1A1 406/4885KDM4E 4465/4885
US-11999754-B2 Ruthenium complexes and their use in olefin metathesis reactions ADH1A, CYP2E1, OPRM1 TRPV1 3365/4885ALDH1A1 78/4885KDM4E 4806/4885
US-20240076308-A1 PROCESS FOR PRODUCING RUTHENIUM COMPLEXES AND INTERMEDIATES THEREOF AND THEIR USE IN OLEFIN METATHESIS POR, CYP1B1, CYP4F11 TRPV1 3244/4885ALDH1A1 406/4885KDM4E 4465/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.