SCHEMBL5960261

SCHEMBL5960261

COC(=O)CC(C)(C)OC(=O)c1ccc2cc(B(O)O)[nH]c2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HTT P42858 2/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KIF11 P52732 2/20 0.34
NPC1 O15118 2/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
HSD17B10 Q99714 3/20 0.33
PKM P14618 2/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24671629 0.81 KIF11 (0.49) RAB9AKDM4EALDH1A1HTTLMNA
SCHEMBL29954766 0.81 KIF11 (0.49) RAB9AKDM4EALDH1A1HTTLMNA
SCHEMBL19463191 0.79 GABRA1 (0.36) RAB9AGABRA1GABRG2GABRB3GABRA3
SCHEMBL29955256 0.71 CREBBP (0.48) RAB9AKDM4EALDH1A1HTTLMNA
SCHEMBL5016542 0.69 KDM4E (0.37) RAB9AKDM4EALDH1A1LMNANPC1
SCHEMBL8479941 0.68 GABRA1 (0.47) RAB9AKDM4EALDH1A1HTTLMNA
SCHEMBL20612118 0.65 RAB9A (0.48) RAB9AKDM4EALDH1A1HTTLMNA
SCHEMBL11888497 0.65 ALDH1A1 (0.53) KDM4EALDH1A1KMT2AMEN1HSD17B10
SCHEMBL3359679 0.65 HRH3 (0.58) RAB9AKDM4EALDH1A1HTTLMNA
SCHEMBL1615765 0.64 GABRA1 (0.46) RAB9AKDM4EALDH1A1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682553-A1 THIENOPYRAZOLES Aventis Pharmaceuticals Inc. (US) 2006-07-26 EP disclosed
WO-2005026175-A1 THIENOPYRAZOLES AVENTIS PHARMACEUTICALS INC. (US) 2005-03-24 WO disclosed