SCHEMBL6002919

SCHEMBL6002919

Cc1cc(Oc2ccnc3ccc(OCCO)cc23)c(-c2ncccn2)nc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.38
MAOA P21397 1/20 0.38
TGFBR1 P36897 8/20 0.36
PDE2A O00408 1/20 0.36
PDE10A Q9Y233 1/20 0.36
DDR2 Q16832 1/20 0.35
SRC P12931 4/20 0.35
BTK Q06187 2/20 0.34
TLR8 Q9NR97 1/20 0.34
AURKA O14965 1/20 0.34
LCK P06239 1/20 0.34
LYN P07948 1/20 0.34
MET P08581 1/20 0.34
FLT1 P17948 1/20 0.34
KDR P35968 1/20 0.34
TEK Q02763 1/20 0.34
AURKB Q96GD4 1/20 0.34
EGFR P00533 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6002895 0.89 TGFBR1 (0.48) SLC22A12MAOATGFBR1PDE2APDE10A
SCHEMBL6004922 0.87 SLC22A12 (0.39) SLC22A12MAOATGFBR1PDE2APDE10A
SCHEMBL6004895 0.85 CYP3A4 (0.45) MAOAALDH1A1HSD17B10
SCHEMBL6004067 0.83 SLC22A12 (0.38) SLC22A12MAOADDR2BTKAURKA
SCHEMBL6005361 0.83 TGFBR1 (0.38) TGFBR1SRCKDRALDH1A1CASP1
SCHEMBL6005251 0.82 PDE2A (0.39) SLC22A12TGFBR1PDE2APDE10ADDR2
SCHEMBL6005388 0.81 TGFBR1 (0.48) MAOATGFBR1TLR8MET
SCHEMBL6004204 0.80 TGFBR1 (0.39) TGFBR1SRC
SCHEMBL3897482 0.77 SRC (0.55) TGFBR1SRCEGFR
SCHEMBL6004343 0.76 SIGMAR1 (0.36) MAOAPDE2APDE10ADDR2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed