SCHEMBL6002895

SCHEMBL6002895

Cc1cc(Oc2ccnc3ccc(OCCO)cc23)c(-c2ccccn2)nc1C

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 13/20 0.48
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
SLC22A12 Q96S37 1/20 0.37
MAOA P21397 1/20 0.36
PDE2A O00408 1/20 0.36
PDE10A Q9Y233 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ACSS2 Q9NR19 1/20 0.35
SRC P12931 2/20 0.34
CBFB Q13951 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6005388 0.92 TGFBR1 (0.48) TGFBR1KDM4ENPC1MAOA
SCHEMBL6002919 0.89 SLC22A12 (0.38) TGFBR1SLC22A12MAOAPDE2APDE10A
SCHEMBL6005265 0.87 TGFBR1 (0.44) TGFBR1KDM4ENPC1SLC22A12MAOA
SCHEMBL6004185 0.87 TGFBR1 (0.59) TGFBR1KDM4ENPC1
SCHEMBL6004274 0.86 TGFBR1 (0.48) TGFBR1KDM4ENPC1MAOA
SCHEMBL3903240 0.85 TGFBR1 (0.49) TGFBR1SRC
SCHEMBL6004761 0.85 TGFBR1 (0.49) TGFBR1SRC
SCHEMBL6005291 0.85 TGFBR1 (0.48) TGFBR1KDM4ENPC1SRC
SCHEMBL6004725 0.84 TGFBR1 (0.48) TGFBR1KDM4ENPC1SRCCBFB
SCHEMBL6004207 0.84 CYP1A2 (0.37) TGFBR1KDM4ENPC1SLC22A12CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed