SCHEMBL6004274

SCHEMBL6004274

Cc1cc(Oc2ccnc3ccc(OCc4ccccc4)cc23)c(-c2ccccn2)nc1C

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 10/20 0.48
CYP3A4 P08684 1/20 0.43
IP6K1 Q92551 1/20 0.40
MAOA P21397 1/20 0.39
NMT1 P30419 1/20 0.38
DYRK1A Q13627 1/20 0.38
MEN1 O00255 1/20 0.38
HSP90AA1 P07900 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
PLAU P00749 1/20 0.37
PLAT P00750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004931 0.92 TGFBR1 (0.48) TGFBR1CYP3A4MAOADYRK1AMEN1
SCHEMBL6004895 0.90 CYP3A4 (0.45) CYP3A4IP6K1MAOANMT1DYRK1A
SCHEMBL6004827 0.87 CYP3A4 (0.44) TGFBR1CYP3A4IP6K1MAOANMT1
SCHEMBL6004185 0.87 TGFBR1 (0.59) TGFBR1MEN1KMT2AKDM4ENPC1
SCHEMBL6002895 0.86 TGFBR1 (0.48) TGFBR1MAOAKDM4ENPC1
SCHEMBL6002971 0.85 ATM (0.49) TGFBR1
SCHEMBL3893031 0.85 ATM (0.49) TGFBR1
SCHEMBL6004725 0.84 TGFBR1 (0.48) TGFBR1KDM4ENPC1
SCHEMBL6004710 0.84 CYP3A4 (0.42) CYP3A4IP6K1NMT1KDM4ENPC1
SCHEMBL6002965 0.84 TGFBR1 (0.49) TGFBR1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed