SCHEMBL6004710

SCHEMBL6004710

CCc1ccc(Oc2ccnc3ccc(OCc4ccccc4)cc23)c(-c2ccccn2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
IP6K1 Q92551 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MET P08581 1/20 0.37
KDR P35968 1/20 0.37
MST1R Q04912 1/20 0.37
PLAU P00749 1/20 0.37
PLAT P00750 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ACSS2 Q9NR19 1/20 0.36
NMT2 O60551 1/20 0.36
NMT1 P30419 1/20 0.36
F2RL3 Q96RI0 1/20 0.36
CBFB Q13951 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004179 0.90 CYP3A4 (0.44) CYP3A4IP6K1KDM4EALDH1A1CYP1A2
SCHEMBL6004827 0.89 CYP3A4 (0.44) CYP3A4IP6K1KDM4EALDH1A1CYP1A2
SCHEMBL6004207 0.87 CYP1A2 (0.37) KDM4EALDH1A1CYP1A2CYP2C9HPGD
SCHEMBL6004082 0.85 CBFB (0.37) KDM4EALDH1A1HPGDHSD17B10MET
SCHEMBL6005438 0.84 MET (0.35) KDM4EALDH1A1HPGDHSD17B10MET
SCHEMBL6004274 0.84 TGFBR1 (0.48) CYP3A4IP6K1KDM4EPLAUPLAT
SCHEMBL6004984 0.83 PDE3B (0.39) KDM4EALDH1A1HPGDHSD17B10MET
SCHEMBL6004857 0.82 SRC (0.37) KDM4EALDH1A1HPGDHSD17B10MET
SCHEMBL6004800 0.80 KDR (0.40) KDM4EALDH1A1HPGDMETKDR
SCHEMBL6002914 0.80 PDGFRB (0.49) METKDRMST1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed