SCHEMBL6004750

SCHEMBL6004750

Cc1csc2ncnc(Oc3cc4cccnc4nc3-c3ccccc3)c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 6/20 0.53
LMNA P02545 3/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
HTT P42858 2/20 0.40
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
DAPK3 O43293 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
ABL1 P00519 1/20 0.34
NTRK1 P04629 1/20 0.34
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004312 0.83 MRGPRX1 (0.56) MRGPRX1LMNACRHBPCRHR2HTT
SCHEMBL6004268 0.81 ALDH1A1 (0.58) MRGPRX1LMNACRHBPCRHR2HTT
SCHEMBL6005337 0.77 ALDH1A1 (0.38) HTTALDH1A1ADORA2AADORA1MET
SCHEMBL13605215 0.72 LCK (0.49) LCKCSF1RRETMETPDGFRB
SCHEMBL6004712 0.72 PRNP (0.43) LMNAHTTALDH1A1HPGDSMN1; SMN2
SCHEMBL6003009 0.72 MAT2A (0.43) LMNAALDH1A1HPGDSMN1; SMN2CYP1A2
SCHEMBL6004877 0.71 KDM4E (0.46) LMNAALDH1A1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL28261532 0.70 PDE10A (0.59) LMNAHTTALDH1A1HPGDRAB9A
SCHEMBL6005342 0.68 MET (0.42) ADORA2AADORA1METPDGFRBPDGFRA
SCHEMBL6004765 0.67 FGFR2 (0.45) PDGFRBPDGFRAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed