SCHEMBL600789

SCHEMBL600789

CCOC(=O)c1cnc(N)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 7/20 0.49
GABRG2 P18507 7/20 0.49
GABRB3 P28472 7/20 0.49
GABRA5 P31644 7/20 0.49
GABRA3 P34903 7/20 0.49
GABRA2 P47869 7/20 0.49
GABRA4 P48169 7/20 0.49
GABRA6 Q16445 7/20 0.49
GABRP O00591 6/20 0.49
GABRD O14764 6/20 0.49
GABRB1 P18505 6/20 0.49
GABRB2 P47870 6/20 0.49
GABRE P78334 6/20 0.49
GABRG1 Q8N1C3 6/20 0.49
GABRG3 Q99928 6/20 0.49
GABRQ Q9UN88 6/20 0.49
ALDH1A1 P00352 4/20 0.49
MAPT P10636 3/20 0.49
NPC1 O15118 3/20 0.49
MEN1 O00255 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31285451 1.00 GABRA1 (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1019601 0.89 CYP1A2 (0.59) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1644521 0.81 POLB (0.70) ALDH1A1KMT2APOLBCYP1A2LMNA
SCHEMBL1644378 0.81 CYP1A2 (0.52) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1020342 0.81 KDM4E (0.50) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL197360 0.80 CYP1A2 (0.50) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL544241 0.79 MAPK1 (0.52) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12184767 0.79 POLB (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL30445565 0.79 POLB (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12986652 0.79 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 111 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026098667-A1 USP30 INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION, PREPARATION METHOD THEREFOR, AND USE THEREOF 长春金赛药业有限责任公司 2026-05-15 WO disclosed
EP-4695252-A1 IMIDAZO[1,2-A]PYRAZINE DERIVATIVES Syngenta Crop Protection AG (CH) 2026-02-18 EP disclosed
WO-2024213659-A1 IMIDAZO[1,2-A]PYRAZINE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2024-10-17 WO disclosed
CN-118684631-A External nucleotide pyrophosphatase/phosphodiesterase 1 (ENPP 1) inhibitors, compositions and uses thereof 中国科学院上海药物研究所 2024-09-24 CN disclosed
CN-113264921-B Pyrazolyl-ureas as kinase inhibitors 瑞斯比维特有限公司 2024-09-13 CN disclosed
US-11724987-B2 Compositions and methods of treating retinal disease ALDEYRA THERAPEUTICS, INC. (US) 2023-08-15 US disclosed
US-11724987-B2 Compositions and methods of treating retinal disease ALDEYRA THERAPEUTICS, INC. (US) 2023-08-15 US disclosed
US-20230091047-A1 FUSED RING PYRIMIDONE DERIVATIVES FOR USE IN THE TREATMENT OF HBV INFECTION OR OF HBV-INDUCED DISEASES JANSSEN PHARMACEUTICA NV (BE) 2023-03-23 US disclosed
US-20230041335-A1 COMPOSITIONS AND METHODS OF TREATING RETINAL DISEASE ALDEYRA THERAPEUTICS, INC. 2023-02-09 US disclosed
EP-3938362-A1 FUSED RING PYRIMIDONE DERIVATIVES FOR USE IN THE TREATMENT OF HBV INFECTION OR OF HBV-INDUCED DISEASES Janssen Sciences Ireland Unlimited Company (IE) 2022-01-19 EP disclosed
EP-2379513-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-10-26 EP disclosed
US-7973025-B2 Compositions and methods of treating retinal disease NEURON SYSTEMS, INC. (US) 2011-07-05 US disclosed
WO-2010078408-A1 HETEROARYL COMPOUNDS USEFUL AS RAF KINASE INHIBITORS BIOGEN IDEC MA INC. (US) 2010-07-08 WO disclosed
EP-1268443-B1 2-HYDROXY-MUTILIN CARBAMATE DERIVATIVES FOR ANTIBACTERIAL USE SMITHKLINE BEECHAM PLC (GB) 2009-07-29 EP disclosed
US-20090182009-A1 Compositions and methods of treating retinal disease NEURON SYSTEMS, INC. (US) 2009-07-16 US disclosed
US-20070135481-A1 Compositions and methods of treating retinal disease ALDEYRA THERAPEUTICS, INC. (F/K/A ALDEXA THERAPEUTICS, INC. F/K/A NEURON SYSTEMS, INC.) 2007-06-14 US disclosed
US-6972297-B2 2-Hydroxy-mutilin carbamate derivatives for antibacterial use SMITHKLINE BEECHAM P.L.C. (GB) 2005-12-06 US disclosed
US-20030114674-A1 2-Hydroxy-mutilin carbamate derivatives for antibacterial use SMITHKLINE BEECHAM P.L.C. (GB) 2003-06-19 US disclosed
EP-1268443-A1 2-HYDROXY-MUTILIN CARBAMATE DERIVATIVES FOR ANTIBACTERIAL USE SmithKline Beecham p.l.c. (GB) 2003-01-02 EP disclosed
WO-2001074788-A1 2-HYDROXY-MUTILIN CARBAMATE DERIVATIVES FOR ANTIBACTERIAL USE SMITHKLINE BEECHAM PLC (GB) 2001-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114674-A1 2-Hydroxy-mutilin carbamate derivatives for antibacterial use MSH6, MSH2, PMS2 GABRA1 1266/4885GABRG2 699/4885GABRB3 1550/4885
US-20230041335-A1 COMPOSITIONS AND METHODS OF TREATING RETINAL DISEASE ALDH1A2, PLA2G2E, CLN6 GABRA1 4108/4885GABRG2 3873/4885GABRB3 3144/4885
US-20230091047-A1 FUSED RING PYRIMIDONE DERIVATIVES FOR USE IN THE TREATMENT OF HBV INFECTION OR OF HBV-INDUCED DISEASES HAVCR2, HCCS, TYMP GABRA1 797/4885GABRG2 523/4885GABRB3 233/4885
US-20090182009-A1 Compositions and methods of treating retinal disease ALDH1A2, PLA2G2E, CLN6 GABRA1 4108/4885GABRG2 3873/4885GABRB3 3144/4885
US-11724987-B2 Compositions and methods of treating retinal disease ALDH1A2, PLA2G2E, CLN6 GABRA1 4108/4885GABRG2 3873/4885GABRB3 3144/4885
US-20070135481-A1 Compositions and methods of treating retinal disease ALDH1A2, PLA2G2E, CLN6 GABRA1 4108/4885GABRG2 3873/4885GABRB3 3144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.