SCHEMBL6008513

SCHEMBL6008513

CC([NH])NS(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.64
SLC1A3 P43003 1/20 0.55
SLC1A2 P43004 1/20 0.55
SLC1A1 P43005 1/20 0.55
ATM Q13315 1/20 0.54
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
PKM P14618 1/20 0.51
PKLR P30613 1/20 0.51
LARS1 Q9P2J5 1/20 0.51
LMNA P02545 3/20 0.50
F2 P00734 2/20 0.50
HSD11B1 P28845 1/20 0.50
CYP19A1 P11511 1/20 0.50
PRSS1 P07477 1/20 0.50
PRSS2 P07478 1/20 0.50
PRSS3 P35030 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
HTR7 P34969 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692936 0.88 L3MBTL1 (0.66) L3MBTL1SLC1A3SLC1A2SLC1A1ATM
SCHEMBL3692115 0.82 L3MBTL1 (0.58) L3MBTL1SLC1A3SLC1A2SLC1A1ATM
SCHEMBL9942084 0.82 ALDH1A1 (0.60) L3MBTL1SLC1A3SLC1A2SLC1A1ATM
SCHEMBL8319592 0.81 SLC1A3 (0.57) L3MBTL1SLC1A3SLC1A2SLC1A1ATM
SCHEMBL7322447 0.81 ADAMTS4 (0.66) L3MBTL1SLC1A3SLC1A2SLC1A1MEN1
SCHEMBL10830548 0.81 ADAMTS4 (0.66) L3MBTL1SLC1A3SLC1A2SLC1A1MEN1
SCHEMBL8905441 0.80 LMNA (0.55) L3MBTL1ATMMEN1KMT2APKM
SCHEMBL20869721 0.80 L3MBTL1 (0.60) L3MBTL1SLC1A3SLC1A2SLC1A1ATM
SCHEMBL6006457 0.80 L3MBTL1 (0.55) L3MBTL1SLC1A3SLC1A2SLC1A1ATM
SCHEMBL10830564 0.80 SLC1A3 (0.56) L3MBTL1SLC1A3SLC1A2SLC1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1207161-B1 NOVEL ISOINDOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2006-01-18 EP disclosed
US-6777410-B2 SUCH AS 9-(2-METHOXYPHENYL)-3-(1-METHYLETHYL)-(1,3)OXAZOLO-(2,3)ISOINDOLE-2,5(3H,9H)-DIONE; DIABETES AND COMPLICATIONS; OBESITY BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-08-17 US disclosed
US-20040053923-A1 Novel isoindole derivatives BANYU PHARMACEUTICAL CO., LTD. 2004-03-18 US disclosed
US-6608098-B1 Diabetes or obesity, 2-(4-(3-isopropyl-2,5-dioxo-2,3-dihydro-1H-pyrrolo(2,1-a) isoindol-9(5H)-yl)phenoxy)-N-propylacetamide BANYU PHARMACEUTICAL CO., LTD. (JP) 2003-08-19 US disclosed
EP-1207161-A1 NOVEL ISOINDOLE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 2002-05-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040053923-A1 Novel isoindole derivatives GPR119, SLC5A2, SLC5A1 L3MBTL1 4136/4885SLC1A3 2390/4885SLC1A2 2008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.