SCHEMBL6015874

SCHEMBL6015874

OCCOc1ccc2[c]c[nH]c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
PDE3B Q13370 3/20 0.40
PDE3A Q14432 3/20 0.40
P2RY12 Q9H244 3/20 0.40
ALDH1A1 P00352 1/20 0.39
RECQL P46063 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
NR1I2 O75469 2/20 0.37
PRKAB2 O43741 4/20 0.36
PRKAG1 P54619 4/20 0.36
PRKAA2 P54646 4/20 0.36
PRKAA1 Q13131 4/20 0.36
PRKAG3 Q9UGI9 4/20 0.36
PRKAG2 Q9UGJ0 4/20 0.36
PRKAB1 Q9Y478 4/20 0.36
TUBB4A P04350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016024 0.81 MAOA (0.36) MAOACYP3A4
SCHEMBL6015813 0.80 KEAP1 (0.46) MAOAALDH1A1PARP1
SCHEMBL6345184 0.80 HPGD (0.47) PDE3BPDE3AALDH1A1CYP3A4SMN1; SMN2
SCHEMBL6015768 0.79 KDM4E (0.47) MAOAALDH1A1PARP1SMN1; SMN2
SCHEMBL6015910 0.78 PDE3B (0.49) PDE3BPDE3AP2RY12ALDH1A1PDE2A
SCHEMBL6015858 0.77 TDP1 (0.33)
SCHEMBL6016063 0.76 LTA4H (0.55)
SCHEMBL6015872 0.76 LTA4H (0.55)
SCHEMBL4602254 0.75 ALOX5 (0.50) MAOAALDH1A1GAASMN1; SMN2
SCHEMBL7620982 0.75 HTR1A (0.42) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed