SCHEMBL6016015

SCHEMBL6016015

COCCNCc1ccc2c(C=O)c[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 2/20 0.53
MAPT P10636 1/20 0.53
CYP2A6 P11509 2/20 0.47
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
PLG P00747 1/20 0.42
PLAU P00749 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
IMPDH2 P12268 1/20 0.41
HTR2A P28223 8/20 0.39
KMT2A Q03164 1/20 0.37
PYGL P06737 1/20 0.37
HTR6 P50406 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015755 0.80 TERT (0.46) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL6819310 0.76 CYP2A6 (0.58) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL29957436 0.76 CYP2A6 (0.58) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL23725271 0.73 CYP2A6 (0.63) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL29152827 0.72 CYP2A6 (0.54) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL6015936 0.72 L3MBTL1 (0.48) CYP2A6L3MBTL1KMT2AMAPK1
SCHEMBL27601642 0.72 ALDH1A1 (0.53) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL7487153 0.71 CYP2A6 (0.57) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL29954469 0.70 ALDH1A1 (1.00) ALDH1A1KDM4EMAPTCYP2A6CYP1A2
SCHEMBL671759 0.70 ALDH1A1 (1.00) ALDH1A1KDM4EMAPTCYP2A6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed