SCHEMBL6015755

SCHEMBL6015755

CN(C)CCCNCc1ccc2c(C=O)c[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TERT O14746 2/20 0.46
CCNA2 P20248 1/20 0.46
CDK2 P24941 1/20 0.46
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
CYP2A6 P11509 2/20 0.45
PLG P00747 1/20 0.40
PLAU P00749 1/20 0.40
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
IMPDH2 P12268 1/20 0.39
SLC6A4 P31645 1/20 0.39
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTR6 P50406 1/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016015 0.80 ALDH1A1 (0.53) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL29957436 0.74 CYP2A6 (0.58) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL6819310 0.74 CYP2A6 (0.58) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL27620200 0.72 ALDH1A1 (0.44) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL15323817 0.72 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL23725271 0.71 CYP2A6 (0.63) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL6015645 0.71 TERT (0.44) TERTCCNA2CDK2KDM4E
SCHEMBL6142482 0.70 TERT (0.46) TERTCCNA2CDK2CYP1A2CYP2C19
SCHEMBL7487153 0.69 CYP2A6 (0.57) ALDH1A1KDM4EMAPTCYP2A6PLG
SCHEMBL16264664 0.68 TERT (0.50) TERTCCNA2CDK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed