SCHEMBL6017539

SCHEMBL6017539

N#CCC1C=CN=C(NCCc2ccc(Oc3ccccc3)cc2)N1c1nc2ccccc2s1.N#CCC1C=CN=C(NCCc2ccccc2Oc2ccccc2)N1c1nc2ccccc2s1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
LTA4H P09960 5/20 0.33
EPHX2 P34913 2/20 0.33
KCNH2 Q12809 3/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NPY1R P25929 1/20 0.31
FES P07332 1/20 0.30
FGFR1 P11362 1/20 0.30
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4192274 0.95 NPC1 (0.31) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL4191147 0.94 RAB9A (0.39) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL7704487 0.90 LTA4H (0.36) LMNALTA4HEPHX2
SCHEMBL4192472 0.86 NPC1 (0.46) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL4186370 0.86 RAB9A (0.42) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL4192264 0.85 LMNA (0.40) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL4190281 0.83 ALDH1A1 (0.40) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL7704544 0.83 ILK (0.41) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL4185618 0.83 KMT2A (0.42) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL4190183 0.83 MAPT (0.40) NPC1RAB9AALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696909-A1 BENZOTHIAZOLE DERIVATIVES FOR THE TREATMENT OF DIABETES Applied Research Systems ARS Holding N.V. (AN) 2006-09-06 EP disclosed
WO-2005025567-A1 BENZOTHIAZOLE DERIVATIVES FOR THE TREATMENT OF DIABETES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2005-03-24 WO disclosed