SCHEMBL6018618

SCHEMBL6018618

Cc1ccc(CNC(=O)c2nc(-c3ccc(F)cc3S(C)(=O)=O)[nH]c(=O)c2CO)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.40
WDR5 P61964 5/20 0.38
ERCC1 P07992 1/20 0.38
FEN1 P39748 1/20 0.38
ERCC4 Q92889 1/20 0.38
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878304 0.94 PTGES (0.42) PTGESWDR5ERCC1FEN1ERCC4
SCHEMBL6885131 0.90 ERCC1 (0.46) PTGESERCC1FEN1ERCC4
SCHEMBL6885310 0.82 PTGES (0.36) PTGESWDR5
SCHEMBL6883870 0.78 EZH2 (0.39) PTGESWDR5CNR1CNR2
SCHEMBL6018615 0.77 KCNE1 (0.44) WDR5CNR1CNR2
SCHEMBL6878399 0.75 PTGES (0.49) PTGESERCC1FEN1ERCC4
SCHEMBL6883711 0.74 NAMPT (0.35) ERCC1FEN1ERCC4
SCHEMBL6883761 0.73 PDE2A (0.38) WDR5ERCC1FEN1ERCC4
SCHEMBL6884265 0.73 WDR5 (0.40) WDR5
SCHEMBL6883027 0.71 PTGES (0.41) PTGESCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037908-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2006-05-02 US disclosed
US-20040229892-A1 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex BRISTOL-MYERS SQUIBB COMPANY 2004-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229892-A1 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex DUT, CDK6, TYMS PTGES 4285/4885WDR5 804/4885ERCC1 2446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.