SCHEMBL5247685

SCHEMBL5247685

O=C(NCCCCCNCCc1ccc(O)cc1)NCCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 4/20 0.37
OPRM1 P35372 4/20 0.37
OPRD1 P41143 3/20 0.37
TRPV1 Q8NER1 1/20 0.35
SLC6A5 Q9Y345 4/20 0.35
GRIA1 P42261 2/20 0.35
ADRB2 P07550 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CHRM1 P11229 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
DRD1 P21728 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
ADRA1A P35348 1/20 0.35
PTGS2 P35354 1/20 0.35
HRH1 P35367 1/20 0.35
DRD3 P35462 1/20 0.35
SLC6A3 Q01959 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6022322 0.85 ADRB2 (0.35) OPRK1OPRM1OPRD1ADRB2ADORA3
SCHEMBL5281472 0.85 TAAR1 (0.37) CHRM1
SCHEMBL6027362 0.85 TRPV1 (0.39) OPRK1OPRM1OPRD1TRPV1SLC6A5
SCHEMBL5805321 0.84 HDAC3 (0.40) TRPV1SLC6A5
SCHEMBL6022468 0.83 ADRB2 (0.43) OPRK1TRPV1ADRB2ADORA3CHRM1
SCHEMBL6027475 0.83 TRPV1 (0.37) OPRK1OPRM1OPRD1TRPV1SLC6A5
SCHEMBL5243798 0.83 FAAH (0.38) TRPV1DRD1ADRA1ADRD3
SCHEMBL6027281 0.82 PDCD1 (0.37) SLC6A5
SCHEMBL6027383 0.81 OPRM1 (0.36) OPRK1OPRM1OPRD1SLC6A5SLC6A2
SCHEMBL6023018 0.81 SLC6A5 (0.38) OPRK1OPRM1OPRD1TRPV1SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856049-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2007-11-21 EP claimed
WO-2006099031-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO claimed