SCHEMBL6024263

SCHEMBL6024263

O=CN(O)CC(Cc1ccc(Cl)c(Cl)c1)C(=O)NNC(=O)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
SIGMAR1 Q99720 2/20 0.43
TRPV1 Q8NER1 1/20 0.40
BMP1 P13497 1/20 0.40
MMP12 P39900 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMO O15229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6024269 0.88 ALDH1A1 (0.48) MEN1KMT2ABMP1MMP12ALDH1A1
SCHEMBL6024223 0.85 HTT (0.45) HTTMEN1KMT2AALDH1A1
SCHEMBL6024204 0.80 BMP1 (0.48) HTTMEN1KMT2ABMP1MMP12
SCHEMBL6024311 0.79 KMO (0.38) HTTMEN1KMT2ASIGMAR1TRPV1
SCHEMBL6024256 0.79 ALDH1A1 (0.52) MEN1KMT2ABMP1ALDH1A1
SCHEMBL3895767 0.76 PNMT (0.42) KMO
SCHEMBL6023703 0.75 BMP1 (0.56) MEN1KMT2ABMP1MMP12
SCHEMBL6024707 0.75 BMP1 (0.56) MEN1KMT2ABMP1MMP12
SCHEMBL6023383 0.75 EPHX2 (0.43) MEN1KMT2AALDH1A1
SCHEMBL6024592 0.74 KMT2A (0.48) MEN1KMT2ABMP1MMP12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363873-B1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2016-04-20 EP claimed
US-7019003-B2 Peptide deformylase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2006-03-28 US claimed
US-20040087585-A1 Peptide deformylase inhibitors GLAXOSMITHKLINE LLC 2004-05-06 US claimed
EP-1363873-B1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2016-04-20 EP disclosed
US-7019003-B2 Peptide deformylase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2006-03-28 US disclosed
EP-1363873-A4 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2006-01-04 EP disclosed
US-20040087585-A1 Peptide deformylase inhibitors GLAXOSMITHKLINE LLC 2004-05-06 US disclosed
EP-1363873-A2 PEPTIDE DEFORMYLASE INHIBITORS SmithKline Beecham Corporation (US) 2003-11-26 EP disclosed
WO-2002070541-A2 PEPTIDE DEFORMYLASE INHIBITORS SMITH KLINE BEECHAM CORPORATION (US) 2002-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087585-A1 Peptide deformylase inhibitors PDF, DPEP1, PEPD HTT 2719/4885MEN1 2224/4885KMT2A 3452/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.