SCHEMBL6044676

SCHEMBL6044676

CCC(C)OC(=O)C(Cc1c[nH]c2ccccc12)(NC=O)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
MAPT P10636 3/20 0.44
POLB P06746 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
APAF1 O14727 1/20 0.44
RECQL P46063 1/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALOX15 P16050 1/20 0.43
TACR3 P29371 2/20 0.42
PKM P14618 1/20 0.41
TACR1 P25103 2/20 0.41
CTSL P07711 1/20 0.40
NMBR P28336 1/20 0.40
ACE P12821 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL837439 0.85 HTT (0.35) KDM4EMAPTL3MBTL1TACR3ALDH1A1
SCHEMBL837267 0.85 NR4A2 (0.39) KDM4EMAPTL3MBTL1TACR1ALDH1A1
SCHEMBL837254 0.85 MPO (0.40) KDM4EMAPTL3MBTL1TACR1ALDH1A1
SCHEMBL837920 0.84 MTNR1A (0.45) KDM4EMAPTL3MBTL1TACR1ALDH1A1
SCHEMBL838321 0.80 PKM (0.55) KDM4EMAPTKMT2AMEN1PKM
SCHEMBL837467 0.76 SPR (0.30)
SCHEMBL4234106 0.74 GPR84 (0.39) KDM4EMAPTPOLBRECQLKMT2A
SCHEMBL4240366 0.74 GPR84 (0.37) KDM4EMAPTPOLBRECQLKMT2A
SCHEMBL4236247 0.72 ALDH1A1 (0.34) KDM4EMAPTPOLBRECQLKMT2A
SCHEMBL8706227 0.70 KDM4E (0.54) KDM4EMAPTPOLBL3MBTL1APAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663184-A2 HYDANTOIN DERIVATIVES AS INHIBITORS OF CELLULAR NECROSIS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2006-06-07 EP disclosed
WO-2005077344-A2 HYDANTOIN DERIVATIVES AS INHIBITORS OF CELLULAR NECROSIS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2005-08-25 WO disclosed