SCHEMBL6047889

SCHEMBL6047889

FC(F)(F)c1cccc(-c2cccc3c2O[C]C3)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.44
HTR7 P34969 1/20 0.44
NOTUM Q6P988 1/20 0.41
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
RORC P51449 1/20 0.39
RORB Q92753 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP11 Q9NR21 1/20 0.39
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
ASIC3 Q9UHC3 1/20 0.38
EPHX2 P34913 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SLC9A1 P19634 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047905 0.90 HTR1A (0.43) HTR1AHTR7NOTUMCHRM2CHRM4
SCHEMBL6047911 0.85 DRD2 (0.46) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4761887 0.75 HTR1A (0.48) HTR1AHTR7NOTUMCHRM2CHRM4
SCHEMBL4596282 0.75 AR (0.37) NOTUMALOX15EPHX2SLC9A1ALDH1A1
SCHEMBL17840165 0.72 RORC (0.57) HTR1AHTR7NOTUMRORCRORB
Ammonia Solution, Strong SCHEMBL27723645 0.71 HTR1A (0.50) HTR1AHTR7NOTUMCHRM2CHRM4
Hydrochloric Acid SCHEMBL3275814 0.69 ASIC3 (0.51) HTR1AHTR7NOTUMPARP10PARP11
SCHEMBL4220301 0.69 PRKAB2 (0.63) HTR1AHTR7NOTUMCHRM2CHRM4
SCHEMBL28667956 0.69 ADORA2A (0.54) HTR7NOTUMRORCRORBEPHX2
SCHEMBL29678302 0.68 TSHR (0.58) NOTUMASIC3ALDH1A1HTR2CKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed