SCHEMBL6067934

SCHEMBL6067934

Nc1nc2ccc(Oc3ccc(F)cc3)cc2s1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.75
NPC1 O15118 4/20 0.75
TP53 P04637 3/20 0.75
SMN1; SMN2 Q16637 3/20 0.75
MAPT P10636 2/20 0.75
HTT P42858 2/20 0.75
AXL P30530 1/20 0.68
GFER P55789 1/20 0.68
CYP3A4 P08684 5/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2C19 P33261 1/20 0.62
HSD17B10 Q99714 3/20 0.61
SCN4A P35499 3/20 0.61
GAA P10253 2/20 0.61
LMNA P02545 2/20 0.61
PKM P14618 2/20 0.61
GMNN O75496 1/20 0.61
USP2 O75604 1/20 0.61
ADORA3 P0DMS8 1/20 0.61
CYP2C9 P11712 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31114771 1.00 RAB9A (0.75) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL20568080 0.90 RAB9A (0.84) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL21186247 0.89 RAB9A (0.68) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL21186277 0.87 RAB9A (0.74) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL7285684 0.86 RAB9A (1.00) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL25306149 0.84 RAB9A (0.75) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL7286497 0.84 CYP3A4 (0.82) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL31114514 0.84 RAB9A (0.75) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL9722831 0.84 RAB9A (0.75) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL7285119 0.84 RAB9A (0.75) RAB9ANPC1TP53SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250382273-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INST NAT SANTE RECH MED (FR) 2025-12-18 US disclosed
EP-4460500-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2024-11-13 EP disclosed
WO-2023131649-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-07-13 WO disclosed
WO-2023131649-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2023-07-13 WO disclosed
WO-2019141980-A1 AGRICULTURAL CHEMICALS GLOBACHEM NV (BE) 2019-07-25 WO disclosed
US-7091227-B2 Benzothiazole derivatives ABBOTT GMBH & CO. KG (DE) 2006-08-15 US disclosed
US-20030153568-A1 Benzothiazole derivatives BASF AKTIENGESELLSCHAFT LUDWIGSHAFEN, GERMANY 2003-08-14 US disclosed
EP-1254123-A1 2-BENZOTHIAZOLYL UREA DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS Abbott GmbH & Co. KG (DE) 2002-11-06 EP disclosed
WO-2001057008-A1 2-BENZOTHIAZOLYL UREA DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS ABBOTT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG & COMPANY KOMMANDITGESELLSCHAFT (DE) 2001-08-09 WO disclosed
EP-0353032-B1 1,5-BENZOTHIAZEPINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CARDIOVASCULAR DISORDERS Sankyo Company Limited (JP) 1992-02-26 EP disclosed
US-5002942-A Calcium channel blockers for cardiovascular disorders SANKYO COMPANY, LIMITED (JP) 1991-03-26 US disclosed
EP-0353032-A1 1,5-benzothiazepine derivatives, their preparation and their use in the treatment of cardiovascular disorders Sankyo Company Limited (JP) 1990-01-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250382273-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS BBOX1, NDUFB6, NDUFB5 RAB9A 2727/4885NPC1 3115/4885TP53 1893/4885
US-20030153568-A1 Benzothiazole derivatives TK1, FLT1, CDK1 RAB9A 3285/4885NPC1 3594/4885TP53 300/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.