SCHEMBL7285684

SCHEMBL7285684

Nc1nc2ccc(Oc3ccccc3)cc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 1.00
TP53 P04637 3/20 1.00
NPC1 O15118 3/20 1.00
SMN1; SMN2 Q16637 2/20 1.00
MAPT P10636 2/20 1.00
HTT P42858 2/20 1.00
L3MBTL1 Q9Y468 2/20 0.68
TDP1 Q9NUW8 1/20 0.68
CYP3A4 P08684 5/20 0.65
CYP1A2 P05177 2/20 0.64
CYP2C19 P33261 1/20 0.64
PI4KA P42356 3/20 0.59
PI4KB Q9UBF8 3/20 0.59
PIK3CA P42336 2/20 0.59
HSD17B10 Q99714 2/20 0.59
SCN4A P35499 2/20 0.59
SCN9A Q15858 2/20 0.59
GAA P10253 2/20 0.59
ALDH1A1 P00352 1/20 0.59
TSHR P16473 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20568080 0.92 RAB9A (0.84) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL11098280 0.87 NPC1 (0.77) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL31114514 0.86 RAB9A (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL6067934 0.86 RAB9A (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL31114771 0.86 RAB9A (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL25306149 0.86 RAB9A (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL7286497 0.86 CYP3A4 (0.82) RAB9ATP53NPC1SMN1; SMN2MAPT
Bromide SCHEMBL11374948 0.86 NPC1 (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL9722831 0.86 RAB9A (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT
SCHEMBL7285119 0.86 RAB9A (0.75) RAB9ATP53NPC1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12629356-B2 Expansion of tumor infiltrating lymphocytes with potassium channel agonists and therapeutic uses thereof IOVANCE BIOTHERAPEUTICS, INC. (US) 2026-05-19 US disclosed
US-12590071-B2 Hydrazone derivative in which terminal amine group is substituted with aryl group or heteroaryl group, and use thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2026-03-31 US disclosed
US-20250382273-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INST NAT SANTE RECH MED (FR) 2025-12-18 US disclosed
EP-3565586-B1 EXPANSION OF TUMOR INFILTRATING LYMPHOCYTES WITH POTASSIUM CHANNEL AGONISTS AND THERAPEUTIC USES THEREOF IOVANCE BIOTHERAPEUTICS INC (US) 2025-10-08 EP disclosed
EP-4570313-A2 CYANOTRIAZOLE COMPOUNDS Otsuka Pharmaceutical Co., Ltd. (JP) 2025-06-18 EP disclosed
CN-113727972-B Novel hydrazone derivatives having terminal amine groups substituted with aryl or heteroaryl groups and use thereof 韩国科学技术研究院 2024-12-27 CN disclosed
EP-4460500-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2024-11-13 EP disclosed
CN-118660885-A Norbornene analogs and their use as potentiators of antitubercular drugs 国家医疗保健研究所 2024-09-17 CN disclosed
WO-2024173715-A1 ANTIFUNGAL COMPOSITIONS AND METHODS OF USE THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2024-08-22 WO disclosed
EP-4219477-A1 CYANOTRIAZOLE COMPOUNDS Otsuka Pharmaceutical Co., Ltd. (JP) 2023-08-02 EP disclosed
US-4994563-A Dyeing, printing cellulose, silk, wool, synthetic polyamides; colorfastness CIBA-GEIGY CORPORATION (US) 1991-02-19 US disclosed
EP-0353032-A1 1,5-benzothiazepine derivatives, their preparation and their use in the treatment of cardiovascular disorders Sankyo Company Limited (JP) 1990-01-31 EP disclosed
EP-0349486-A2 Azo dyes, their preparation and their use CIBA-GEIGY AG (CH) 1990-01-03 EP disclosed
EP-0261459-A2 N-benzothiazolyl amides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1988-03-30 EP disclosed
US-4438126-A Lower alkanoic acid derivatives of 2-oxo-benzoxazolines and aldose reductase inhibiting compositions thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-03-20 US disclosed
EP-0022317-B1 2-OXO-BENZOTHIAZOLINE, BENZOXAZOLINE OR INDOLINE DERIVATIVES, THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-09-21 EP disclosed
US-4370340-A ANTIDIABETIC AGENT FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-01-25 US disclosed
US-4233214-A FOR POLYACRYLONITRILE AND ACID-MODIFIED POLYESTERS OR POLYAMIDES BAYER AKTIENGESELLSCHAFT (DE) 1980-11-11 US disclosed
US-4036826-A Cationic azo dyestuffs with a hydroxyalkylated ammonium group BAYER AKTIENGESELLSCHAFT (DT) 1977-07-19 US disclosed
US-4006127-A Cationic diazacyanine dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1977-02-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12629356-B2 Expansion of tumor infiltrating lymphocytes with potassium channel agonists and therapeutic uses thereof PBK, IL2, KCNN3 RAB9A 4594/4885TP53 291/4885NPC1 1565/4885
US-20250382273-A1 BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS BBOX1, NDUFB6, NDUFB5 RAB9A 2727/4885TP53 1893/4885NPC1 3115/4885
US-12590071-B2 Hydrazone derivative in which terminal amine group is substituted with aryl group or heteroaryl group, and use thereof ABL1, TH, CYP3A43 RAB9A 1131/4885TP53 3499/4885NPC1 1264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.