SCHEMBL6071234

SCHEMBL6071234

COC(=O)CC(Nc1ccccc1OC)c1csc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.41
HTR1D P28221 2/20 0.41
CASP3 P42574 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALOX5 P09917 1/20 0.39
PKM P14618 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
APLNR P35414 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13413859 0.78 IDO1 (0.41) CYP1A2CYP3A4GAACYP2C9CYP2C19
SCHEMBL3306466 0.74 ALDH1A1 (0.49) CYP1A2GAASMN1; SMN2MAPT
SCHEMBL6070968 0.70 MAPT (0.46) CYP1A2CYP3A4GAACYP2C9CYP2C19
SCHEMBL6071098 0.69 RAB9A (0.54) CYP1A2CYP3A4GAACYP2C9SMN1; SMN2
SCHEMBL6070967 0.69 L3MBTL1 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19SMN1; SMN2
SCHEMBL27962281 0.67 ALDH1A1 (0.50) CYP1A2CYP3A4GAACYP2C9CYP2C19
SCHEMBL12971503 0.67 ALOX5 (0.50) HTR1AHTR1DGAAALOX5PKM
SCHEMBL6999400 0.67 ALOX5 (0.54) ALOX5PKMSMN1; SMN2MAPT
SCHEMBL24704555 0.66 CYP2A6 (0.46) SMN1; SMN2TP53
SCHEMBL6071237 0.66 HTR1A (0.41) HTR1AHTR1DCASP3CYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060014752-A1 Heterocyclic anti-epileptogenic agents and methods of use thereof QUEEN'S UNIVERSITY AT KINGSTON (CA) 2006-01-19 US disclosed
US-20030114441-A1 Heterocyclic anti-epileptogenic agents and methods of use thereof QUEEN'S UNIVERSITY AT KINGSTON (CA) 2003-06-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114441-A1 Heterocyclic anti-epileptogenic agents and methods of use thereof CA3, GAP43, SLC1A2 HTR1A 790/4885HTR1D 1804/4885CASP3 1784/4885
US-20060014752-A1 Heterocyclic anti-epileptogenic agents and methods of use thereof GAP43, GABRE, CA3 HTR1A 805/4885HTR1D 1632/4885CASP3 1663/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.