SCHEMBL6078624

SCHEMBL6078624

CC(CCc1ccc(Cl)c(Cl)c1)CC(N)=O

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 6/20 0.47
SIGMAR1 Q99720 5/20 0.47
PNMT P11086 2/20 0.46
TAAR1 Q96RJ0 1/20 0.46
LIPG Q9Y5X9 3/20 0.43
KCNH2 Q12809 5/20 0.42
TSHR P16473 1/20 0.42
PAX8 Q06710 1/20 0.42
PYGL P06737 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16973611 0.80 ALDH1A1 (0.40) TMEM97SIGMAR1KCNH2
SCHEMBL4910377 0.79 PNMT (0.58) TMEM97SIGMAR1PNMTTAAR1KCNH2
SCHEMBL4986765 0.77 PNMT (0.42) TMEM97SIGMAR1PNMTTAAR1LIPG
SCHEMBL661213 0.76 TSHR (0.51) TSHR
SCHEMBL4983954 0.75 PNMT (0.46) TMEM97SIGMAR1PNMTTAAR1LIPG
SCHEMBL10859086 0.75 PNMT (0.67) TMEM97SIGMAR1PNMTTAAR1KCNH2
SCHEMBL14731704 0.75 PNMT (0.67) TMEM97SIGMAR1PNMTTAAR1KCNH2
SCHEMBL3393678 0.75 PYGL (0.57) SIGMAR1PNMTTAAR1TSHRPYGL
SCHEMBL7089879 0.75 ALDH1A1 (0.43)
SCHEMBL12436727 0.75 SIGMAR1 (0.58) TMEM97SIGMAR1PNMTTAAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109186-B2 4-hydroxy-5-oxo-1-(2-[4-methylpiperazin-1-yl]ethyl)-2,5-dihydro-1H-pyrrole-3-carboxylic acid (3,4-dichlorobenzyl)-methyl-amide for human immunodeficiency virus (HIV) treatment BRISTOL-MYERS SQUIBB COMPANY (US) 2006-09-19 US disclosed
US-20040110804-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-06-10 US disclosed
WO-2004004657-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-01-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040110804-A1 HIV integrase inhibitors CDKN1A, SAMHD1, CTCF TMEM97 3926/4885SIGMAR1 4036/4885PNMT 2181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.