SCHEMBL6083117

SCHEMBL6083117

O=c1n(-c2ccc(OCCN3CCN(c4ccccc4)CC3)cc2)ccn1-c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.59
DRD3 P35462 4/20 0.59
HRH1 P35367 3/20 0.59
HTR1A P08908 3/20 0.59
HTR2A P28223 3/20 0.59
TMEM97 Q5BJF2 3/20 0.59
SIGMAR1 Q99720 3/20 0.59
HRH3 Q9Y5N1 3/20 0.58
HRH2 P25021 1/20 0.58
LTA4H P09960 2/20 0.56
MCHR1 Q99705 5/20 0.50
KCNH2 Q12809 2/20 0.50
MCHR2 Q969V1 1/20 0.49
SLC6A2 P23975 2/20 0.49
SLC6A4 P31645 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728674 0.88 ALDH1A1 (0.60) DRD2DRD3HRH1HRH3HRH2
SCHEMBL6081563 0.87 LTA4H (0.55) HRH3LTA4HMCHR1KCNH2MCHR2
SCHEMBL1728438 0.86 LTA4H (0.56) HRH1HRH3HRH2LTA4HMCHR1
SCHEMBL1728604 0.84 DRD3 (0.59) DRD2DRD3SIGMAR1LTA4HMCHR1
SCHEMBL1728503 0.84 LTA4H (0.54) TMEM97SIGMAR1HRH3LTA4HMCHR1
SCHEMBL1728694 0.84 KDM4E (0.56) SIGMAR1HRH3LTA4HMCHR1KCNH2
SCHEMBL1729170 0.82 LTA4H (0.51) HRH1HRH3HRH2LTA4HMCHR1
SCHEMBL1728498 0.82 LTA4H (0.51) HRH1HRH3HRH2LTA4HMCHR1
SCHEMBL6081977 0.81 LTA4H (0.56) DRD2DRD3HRH1HTR1AHTR2A
SCHEMBL6081709 0.81 TMEM97 (0.69) TMEM97SIGMAR1HRH3LTA4HMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed