SCHEMBL6096554

SCHEMBL6096554

O=C1C=C(Cl)C(=O)C(c2c[nH]c3c(Br)cccc23)=C1Cl

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.41
CLK1 P49759 6/20 0.40
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
GSK3B P49841 1/20 0.40
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
AR P10275 3/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
PARP1 P09874 1/20 0.32
SLC6A4 P31645 1/20 0.31
CAMK2D Q13557 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6097786 0.86 DYRK1A (0.43) DYRK1AARAURKAAURKBNR3C1
SCHEMBL6097207 0.84 AR (0.44) AR
SCHEMBL6096052 0.84 GPR84 (0.40) ARAURKAAURKBNR3C1PGR
SCHEMBL6094634 0.82 PARP1 (0.40) CLK1CDK5PIM1ARAURKA
SCHEMBL6095205 0.82 CSNK2A2 (0.41) PIM1ARCAMK2D
SCHEMBL6095726 0.81 ALDH1A1 (0.44) DYRK1AGSK3BARAURKAAURKB
SCHEMBL6096077 0.81 AR (0.35) ARAURKAAURKBNR3C1PGR
SCHEMBL6097186 0.79 MEN1 (0.37) ARNR3C1PGRNR3C2
SCHEMBL6096170 0.79 CYP2A6 (0.41) CLK1CDK5CDK5R1AURKAAURKB
SCHEMBL6097734 0.78 PRKCB (0.54) GSK3BPIM1CAMK2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7057052-B2 Heterocyclic quinones as pharmaceutical agents DUKE UNIVERSITY (US) 2006-06-06 US disclosed
WO-2004050014-A2 SETEROCYCLIC QUINONES AS PHARMACEUTICAL AGENTS DUKE UNIVERSITY (US) 2004-06-17 WO disclosed
US-20040063774-A1 Heterocyclic quinones as pharmaceutical agents DUKE UNIVERSITY 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063774-A1 Heterocyclic quinones as pharmaceutical agents NQO1, RECQL, SDHA DYRK1A 2359/4885CLK1 4001/4885CDK5 88/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.