SCHEMBL6094634

SCHEMBL6094634

O=C1C=C(Cl)C(=O)C(c2c[nH]c3c(-c4ccccc4)cccc23)=C1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
CLK1 P49759 2/20 0.36
CLK2 P49760 2/20 0.36
CLK3 P49761 2/20 0.36
CNR2 P34972 1/20 0.36
FEN1 P39748 1/20 0.36
AR P10275 3/20 0.36
NR3C1 P04150 2/20 0.36
PGR P06401 2/20 0.36
NR3C2 P08235 2/20 0.36
IMPDH2 P12268 2/20 0.35
KDM4E B2RXH2 1/20 0.35
AURKB Q96GD4 2/20 0.34
MAP4K4 O95819 1/20 0.34
CSF1R P07333 1/20 0.34
FGFR1 P11362 1/20 0.34
PDGFRA P16234 1/20 0.34
LTK P29376 1/20 0.34
KDR P35968 1/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6097786 0.84 DYRK1A (0.43) ARNR3C1PGRNR3C2AURKB
SCHEMBL6096554 0.82 DYRK1A (0.41) PARP1CLK1ARNR3C1PGR
SCHEMBL6096052 0.82 GPR84 (0.40) ARNR3C1PGRNR3C2AURKB
SCHEMBL6097207 0.82 AR (0.44) ARKDM4EALDH1A1PRKCBPRKCA
SCHEMBL6095205 0.82 CSNK2A2 (0.41) ARKDM4EPTPRCPTPRFPTPN1
SCHEMBL6096812 0.81 FEN1 (0.39) FEN1PTPN1ALDH1A1SIRT2
SCHEMBL6096077 0.79 AR (0.35) ARNR3C1PGRNR3C2KDM4E
SCHEMBL6095726 0.79 ALDH1A1 (0.44) CNR2ARNR3C1PGRNR3C2
SCHEMBL6097734 0.79 PRKCB (0.54) IMPDH2PTPRCPTPRFPTPN1CDC25B
SCHEMBL6096277 0.78 LTA4H (0.47) IMPDH2SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7057052-B2 Heterocyclic quinones as pharmaceutical agents DUKE UNIVERSITY (US) 2006-06-06 US disclosed
WO-2004050014-A2 SETEROCYCLIC QUINONES AS PHARMACEUTICAL AGENTS DUKE UNIVERSITY (US) 2004-06-17 WO disclosed
US-20040063774-A1 Heterocyclic quinones as pharmaceutical agents DUKE UNIVERSITY 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063774-A1 Heterocyclic quinones as pharmaceutical agents NQO1, RECQL, SDHA PARP1 259/4885CLK1 4001/4885CLK2 3213/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.