SCHEMBL6142202

SCHEMBL6142202

Cc1cccc2nc(C(=O)OC(C)(C)C)[nH]c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GLA P06280 2/20 0.36
BCHE P06276 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
GAA P10253 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340375 0.86 ADRA1A (0.37) KDM4EALDH1A1GLABCHEMEN1
SCHEMBL30831141 0.82 BRPF1 (0.42) KDM4EALDH1A1GLAMEN1KMT2A
SCHEMBL28882676 0.82 BRPF1 (0.42) KDM4EALDH1A1GLAMEN1KMT2A
SCHEMBL10662224 0.81 GAA (0.37) KDM4EALDH1A1GLABCHEMEN1
SCHEMBL9241391 0.80 XDH (0.35) KDM4EALDH1A1PARP1NR4A2HPGD
SCHEMBL1144716 0.79 PIN1 (0.49) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL27552206 0.78 XDH (0.52) KDM4EALDH1A1BCHEMEN1KMT2A
SCHEMBL2475448 0.77 PARP1 (0.40) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL6142201 0.77 HRH4 (0.52) KDM4EALDH1A1GAANPC1RAB9A
SCHEMBL6954527 0.75 GABRA1 (0.35) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944604-B1 GUANIDINYL HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS PROCTER & GAMBLE (US) 2005-01-12 EP disclosed
EP-0944601-B1 GUANIDINYLAMINO HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS PROCTER & GAMBLE (US) 2003-02-12 EP disclosed
EP-0944604-A1 GUANIDINYL HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1999-09-29 EP disclosed
WO-1998023596-A1 GUANIDINYL HETEROCYCLE COMPOUNDS USEFUL AS ALPHA-2 ADRENOCEPTOR AGONISTS THE PROCTER & GAMBLE COMPANY (US) 1998-06-04 WO disclosed