SCHEMBL6153220

SCHEMBL6153220

COc1ccc(N2CCN(c3ccccc3)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.66
PKM P14618 1/20 0.66
MAPT P10636 5/20 0.66
RAB9A P51151 2/20 0.66
KMT2A Q03164 2/20 0.66
HTR3E A5X5Y0 1/20 0.63
HTR3B O95264 1/20 0.63
ADRB1 P08588 1/20 0.63
HTR3A P46098 1/20 0.63
HTR3D Q70Z44 1/20 0.63
HTR3C Q8WXA8 1/20 0.63
SIGMAR1 Q99720 1/20 0.63
DRD2 P14416 1/20 0.61
MAPK1 P28482 1/20 0.59
L3MBTL1 Q9Y468 2/20 0.59
NPSR1 Q6W5P4 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
NPC1 O15118 1/20 0.58
HTR1A P08908 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30277734 0.92 ALDH1A1 (0.58) ALDH1A1PKMMAPTRAB9AKMT2A
SCHEMBL29656856 0.91 HTR3E (0.73) ALDH1A1MAPTRAB9AKMT2AHTR3E
SCHEMBL28599511 0.91 HTR3E (0.73) ALDH1A1MAPTRAB9AKMT2AHTR3E
SCHEMBL19212406 0.84 ADRB1 (0.69) ALDH1A1MAPTRAB9AKMT2AADRB1
SCHEMBL14362730 0.83 HTR3E (0.63) ALDH1A1MAPTRAB9AKMT2AHTR3E
SCHEMBL424503 0.83 DRD2 (0.66) ALDH1A1MAPTRAB9AKMT2AHTR3E
SCHEMBL11396473 0.83 MAPT (0.65) ALDH1A1PKMMAPTRAB9AKMT2A
SCHEMBL11923385 0.83 SIGMAR1 (0.79) ALDH1A1PKMMAPTKMT2ASIGMAR1
SCHEMBL2464580 0.83 ALDH1A1 (0.66) ALDH1A1MAPTRAB9AKMT2ADRD2
SCHEMBL2925759 0.83 HTR3E (0.68) ALDH1A1MAPTRAB9AKMT2AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2721013-B1 PROCESS FOR THE PREPARATION OF A CHIRAL COMPOUND SANDOZ AG (CH) 2018-02-21 EP disclosed
EP-1068200-B1 2,4,4-TRISUBSTITUTED-1,3-DIOXOLANE ANTIFUNGALS JANSSEN PHARMACEUTICA NV (BE) 2005-02-16 EP disclosed
US-6387906-B1 DERMATOPHYTES JANSSEN PHARMACEUTICA N.V. (BE) 2002-05-14 US disclosed
EP-1068200-A1 2,4,4-TRISUBSTITUTED-1,3-DIOXOLANE ANTIFUNGALS JANSSEN PHARMACEUTICA N.V. (BE) 2001-01-17 EP disclosed
WO-1999002523-A1 2,4,4-TRISUBSTITUTED-1,3-DIOXOLANE ANTIFUNGALS JANSSEN PHARMACEUTICA N.V. (BE) 1999-01-21 WO disclosed