SCHEMBL6154529

SCHEMBL6154529

C=CCN(CC=C)c1cccc(C(=O)C(C)(C)CC(=O)OCC)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.42
HSD11B1 P28845 1/20 0.38
ALOX5 P09917 1/20 0.35
HTT P42858 1/20 0.35
MAPT P10636 3/20 0.34
GAA P10253 3/20 0.34
LMNA P02545 2/20 0.34
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPK1 P28482 2/20 0.34
TSHR P16473 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14898280 0.80 LMNA (0.49) PTPN1ALOX5MAPTGAALMNA
SCHEMBL6154598 0.75 HSD11B1 (0.44) HSD11B1LMNAALDH1A1SMN1; SMN2NPC1
SCHEMBL6401663 0.74 HSD11B1 (0.57) HSD11B1MAPTLMNAALDH1A1NPSR1
SCHEMBL876064 0.72 PTPN1 (0.49) PTPN1LMNAALDH1A1KMT2ATSHR
SCHEMBL4876996 0.69 LMNA (0.48) MAPTGAALMNAALDH1A1NPSR1
SCHEMBL611180 0.69 PTPN1 (0.45) PTPN1MAPTALDH1A1KMT2ATSHR
SCHEMBL4872329 0.68 LMNA (0.41) HTTMAPTGAALMNAALDH1A1
SCHEMBL3611806 0.68 ESR1 (0.54) HSD11B1MAPTLMNAALDH1A1KMT2A
SCHEMBL20138852 0.67 KMT2A (0.49) HSD11B1HTTMAPTLMNAALDH1A1
SCHEMBL1470467 0.67 CA12 (0.53) ALOX5HTTMAPTGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
EP-1499603-A1 ANTIVIRAL LACTONE-UREAS Bayer Aktiengesellschaft (DE) 2005-01-26 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed
WO-2003089421-A1 ANTIVIRAL LACTONE-UREAS BAYER HEALTHCARE AG (DE) 2003-10-30 WO disclosed