SCHEMBL6157817

SCHEMBL6157817

O=COC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.53
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
SCN1A P35498 5/20 0.48
SCN2A Q99250 5/20 0.48
SCN3A Q9NY46 5/20 0.48
SLC6A3 Q01959 3/20 0.47
SLC6A4 P31645 2/20 0.47
CHRNB2 P17787 3/20 0.47
CHRNB4 P30926 3/20 0.47
CHRNA3 P32297 3/20 0.47
CHRNA4 P43681 3/20 0.47
HNF4A P41235 1/20 0.46
TSHR P16473 1/20 0.45
RECQL P46063 1/20 0.45
ADORA3 P0DMS8 1/20 0.44
GPR52 Q9Y2T5 1/20 0.43
FABP3 P05413 1/20 0.42
FABP4 P15090 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1901065 0.84 BCAT2 (0.52) BCAT2MEN1KMT2ASMN1; SMN2SCN1A
SCHEMBL5806493 0.82 CYP3A4 (0.47) TSHRPOLB
SCHEMBL9790236 0.80 BCAT2 (0.61) BCAT2MEN1KMT2ASMN1; SMN2SCN1A
SCHEMBL28444799 0.80 BCAT2 (0.61) BCAT2MEN1KMT2ASMN1; SMN2SCN1A
SCHEMBL8662843 0.79 BCAT2 (0.64) BCAT2MEN1KMT2ASMN1; SMN2SCN1A
SCHEMBL2359279 0.79 ALDH1A1 (0.58) SMN1; SMN2TSHRPOLB
SCHEMBL28172838 0.77 HNF4A (0.46) SMN1; SMN2HNF4AFABP3FABP4FABP5
SCHEMBL28366814 0.77 BCAT2 (0.62) BCAT2MEN1KMT2ASMN1; SMN2SCN1A
SCHEMBL3964332 0.77 BCAT2 (0.57) BCAT2MEN1KMT2ASMN1; SMN2SCN1A
SCHEMBL28065469 0.77 BCAT2 (0.57) BCAT2MEN1KMT2ASMN1; SMN2SCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-20040157894-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-08-12 US disclosed
US-6699881-B2 MATRIX METALLOPROTEASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-02 US disclosed
US-20030078253-A1 Thiol compounds, their production and use TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-24 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-1132379-A1 NOVEL THIOL DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND UTILIZATION THEREOF Takeda Chemical Industries, Ltd. (JP) 2001-09-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078253-A1 Thiol compounds, their production and use TST, QSOX1, SULT1E1 BCAT2 1079/4885MEN1 3957/4885KMT2A 1898/4885
US-20040157894-A1 Thiol compounds, their production and use TST, SULT1E1, QSOX1 BCAT2 1168/4885MEN1 3906/4885KMT2A 1850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.