Sulfadoxine

Sulfadoxine

SCHEMBL615997

COc1ncnc(NS(=O)(=O)c2ccc(N)cc2)c1OC.Nc1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPPK-DHPS

The experimentally established mechanism targets of Sulfadoxine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.90
MEN1 O00255 1/20 0.63
KMT2A Q03164 1/20 0.63
CYP2C19 P33261 2/20 0.51
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
HTT P42858 1/20 0.49
CA9 Q16790 1/20 0.49
LMNA P02545 3/20 0.48
CA7 P43166 2/20 0.47
CA13 Q8N1Q1 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
CYP19A1 P11511 1/20 0.44
CCR4 P51679 2/20 0.43
HTR6 P50406 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfadoxine SCHEMBL29390814 0.95 ESR1 (1.00) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL41069 0.95 ESR1 (1.00) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL28436237 0.94 ESR1 (0.97) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL27856131 0.94 ESR1 (0.97) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL28359083 0.94 ESR1 (0.97) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL28537335 0.94 ESR1 (0.97) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL28122268 0.89 ESR1 (0.88) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL30005494 0.88 ESR1 (0.86) ESR1MEN1KMT2ACYP2C19LMNA
Sulfadoxine SCHEMBL28198178 0.86 ESR1 (0.82) ESR1MEN1KMT2ACYP2C19LMNA
Sulfalene SCHEMBL28086248 0.84 MEN1 (0.90) ESR1MEN1KMT2ACYP2C19CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112020562-A CRISPR-Effector System-based diagnostics 博德研究所 2020-12-01 CN disclosed
CN-111836903-A Multiple diagnostics based on CRISPR effector systems 博德研究所 2020-10-27 CN disclosed
CN-111630162-A CRISPR-Effector System-based diagnostics 博德研究所 2020-09-04 CN disclosed
EP-3692367-A1 DIAGNOSTIC MEANS FOR THE DETECTION AND/OR QUANTIFICATION OF A PLURALITY OF ANALYTES PRESENT IN A SAMPLE Unisensor (BE) 2020-08-12 EP disclosed
CN-111448311-A Multi-effector CRISPR-based diagnostic systems 博德研究所 2020-07-24 CN disclosed
CN-111108220-A CRISPR-Effector System-based diagnostics for Virus detection 博德研究所 2020-05-05 CN disclosed
WO-2019068806-A1 DIAGNOSTIC MEANS FOR THE DETECTION AND/OR QUANTIFICATION OF A PLURALITY OF ANALYTES PRESENT IN A SAMPLE UNISENSOR (BE) 2019-04-11 WO disclosed
US-8383154-B2 Swellable dosage form comprising gellan gum EGALET A/S (DK) 2013-02-26 US disclosed
US-8383155-B2 Swellable dosage form comprising gellan gum EGALET A/S (DK) 2013-02-26 US disclosed
US-20120039969-A1 SWELLABLE DOSAGE FORM COMPRISING GELLAN GUM EGALET A/S 2012-02-16 US disclosed
EP-1758557-B1 SWELLABLE DOSAGE FORM COMPRISING GELLAN GUM EGALET LTD (GB) 2011-07-13 EP disclosed
EP-2258349-A2 Swellable dosage form comprising gellan gum Egalet A/S (DK) 2010-12-08 EP disclosed
US-7670631-B2 Method for the prevention of malaria infection of humans by hepatocyte growth factor antagonists ALFAMA—Investigação e Desenvolvimento de Produtos Farmacêuticos, Lda. (PT) 2010-03-02 US disclosed
US-20080299199-A1 Swellable Dosage Form Comprising Gellan Gum EGALET A/S 2008-12-04 US disclosed
EP-1758557-A2 SWELLABLE DOSAGE FORM COMPRISING GELLAN GUM Egalet A/S (DK) 2007-03-07 EP disclosed
EP-1601378-A2 A METHOD FOR THE PREVENTION OF MALARIA INFECTION OF HUMANS BY HEPATOCYTE GROWTH FACTOR ANTAGONISTS Instituto Gulbenkian de Ciencia (PT) 2005-12-07 EP disclosed
WO-2005107713-A2 SWELLABLE DOSAGE FORM COMPRISING GELLAN GUM EGALET A/S (DK) 2005-11-17 WO disclosed
WO-2004080420-A2 A METHOD FOR THE PREVENTION OF MALARIA INFECTION OF HUMANS BY HEPATOCYTE GROWTH FACTOR ANTAGONISTS INSTITUTO GULBENKIAN DE CIENCIA (PT) 2004-09-23 WO disclosed
US-20040185050-A1 Method for the prevention of malaria infection of humans by hepatocyte growth factor antagonists ALFAMA - INVESTIGACAO E DESENVOLVIMENTO DE PRODUTOS FARMACEUTICOS LDA. (PT) 2004-09-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120039969-A1 SWELLABLE DOSAGE FORM COMPRISING GELLAN GUM PUF60, COG6, GP6 ESR1 4843/4885MEN1 1971/4885KMT2A 3976/4885
US-20080299199-A1 Swellable Dosage Form Comprising Gellan Gum GP6, PUF60, SELL ESR1 4796/4885MEN1 2890/4885KMT2A 4038/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.