SCHEMBL6164485

SCHEMBL6164485

N#CCCn1nc(COc2ccccc2)c2c1CCC2=O

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.47
CYP1A2 P05177 2/20 0.37
TSHR P16473 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165037 0.82 MAOB (0.42) MAOBCYP1A2TSHRHIF1A
SCHEMBL6162649 0.74 PARP1 (0.37) MAOBCYP1A2TSHRHIF1A
SCHEMBL6166684 0.72 MAOB (0.33) MAOBCYP1A2TSHR
SCHEMBL6165983 0.71 ATM (0.44) MAOBCYP1A2TSHR
SCHEMBL6163581 0.70 CYP1A2 (0.36) CYP1A2TSHRHIF1A
SCHEMBL6165490 0.70 LMNA (0.49) CYP1A2TSHRHIF1A
SCHEMBL6167954 0.70 HTT (0.32)
SCHEMBL6167036 0.69 RIPK3 (0.39) MAOB
SCHEMBL6166254 0.69 ALDH1A1 (0.38) MAOBTSHRHIF1A
SCHEMBL6164339 0.69 HTT (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed