SCHEMBL6166582

SCHEMBL6166582

Cc1nn(-c2ccc(Cl)nn2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 18/20 0.64
CCNA2 P20248 1/20 0.61
CDK2 P24941 1/20 0.61
OPRK1 P41145 4/20 0.59
OPRD1 P41143 3/20 0.59
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6166153 0.84 CCNA2 (0.47) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6167734 0.84 OPRM1 (0.49) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6165838 0.83 OPRM1 (0.62) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6165095 0.82 ALDH1A1 (0.58) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6162652 0.82 CCNA2 (0.45) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6166409 0.81 OPRM1 (0.56) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6166892 0.78 CCNA2 (0.53) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6164838 0.77 CCNA2 (0.41) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6162861 0.76 OPRM1 (0.65) OPRM1CCNA2CDK2OPRK1OPRD1
SCHEMBL6771820 0.75 OPRM1 (0.75) OPRM1OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed