SCHEMBL6167006

SCHEMBL6167006

O=C(O)c1ccc2c(c1)CN(Cc1ccc(F)c(F)c1)CC2=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HTT P42858 1/20 0.42
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
TSHR P16473 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
HTR2A P28223 1/20 0.39
MCHR1 Q99705 1/20 0.39
PTGER4 P35408 2/20 0.39
HPGD P15428 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HIF1A Q16665 1/20 0.38
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
PTGER2 P43116 1/20 0.37
SRD5A1 P18405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169451 0.87 PTGER4 (0.42) L3MBTL1PTGER4PTGER2POLBMEN1
SCHEMBL6169204 0.86 ACACB (0.43) ALDH1A1HTTS1PR3SIGMAR1POLB
SCHEMBL6168303 0.84 PTGER4 (0.47) ALDH1A1MCHR1PTGER4PTGER2POLB
SCHEMBL6169640 0.80 AR (0.42) ALDH1A1TSHRCYP2D6CYP2C9MEN1
SCHEMBL6168750 0.79 LMNA (0.46) HPGDMEN1KMT2A
SCHEMBL6168074 0.77 RHEB (0.39) PTGER4HPGDPTGER2SRD5A1POLB
SCHEMBL6167129 0.76 XDH (0.43)
SCHEMBL6761908 0.74 KMT2A (0.68) ALDH1A1HPGDPOLBMEN1KMT2A
SCHEMBL2722964 0.71 MEN1 (0.49) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL1684479 0.70 MAPT (0.59) ALDH1A1HTTTSHRL3MBTL1PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530472-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004014379-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed