SCHEMBL6168074

SCHEMBL6168074

CC(C)(C)OC(=O)c1ccc(CN2CC(=O)c3ccc(C(=O)O)cc3C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
SRD5A1 P18405 1/20 0.39
ACACB O00763 3/20 0.38
KDM1A O60341 3/20 0.38
LTA4H P09960 1/20 0.38
PTGER4 P35408 1/20 0.37
PTGER2 P43116 1/20 0.37
ACHE P22303 1/20 0.37
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.36
ENPP2 Q13822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6168750 0.80 LMNA (0.46) ACACBMEN1HPGDKMT2AENPP2
SCHEMBL6169640 0.79 AR (0.42) ACHEMEN1KMT2A
SCHEMBL2722964 0.77 MEN1 (0.49) ACACBMEN1KMT2A
SCHEMBL6167006 0.77 ALDH1A1 (0.42) SRD5A1PTGER4PTGER2MEN1HPGD
SCHEMBL6167129 0.74 XDH (0.43)
SCHEMBL6168895 0.73 CYP3A4 (0.47) ACACBMEN1KMT2A
SCHEMBL25142596 0.72 CHKA (0.61) SIRT2SIRT1KDM1A
SCHEMBL6169204 0.72 ACACB (0.43) ACACBPOLB
SCHEMBL6169451 0.72 PTGER4 (0.42) PTGER4PTGER2MEN1KMT2APOLB
SCHEMBL18173436 0.71 KDM1A (0.46) SIRT2SIRT1KDM1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530472-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004014379-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed