SCHEMBL6169451

SCHEMBL6169451

COc1ccc(C(N)=O)cc1.O=C(O)c1ccc2c(c1)CN(Cc1ccc(F)c(F)c1)CC2=O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.42
PTGER2 P43116 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CCR3 P51677 1/20 0.39
PARP10 Q53GL7 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PARP1 P09874 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
PARP4 Q9UKK3 1/20 0.38
ABCB1 P08183 1/20 0.38
TAS2R14 Q9NYV8 2/20 0.38
GRM2 Q14416 2/20 0.38
OPRM1 P35372 1/20 0.37
CHRM1 P11229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6168303 0.91 PTGER4 (0.47) PTGER4PTGER2POLBMEN1KMT2A
SCHEMBL6167006 0.87 ALDH1A1 (0.42) PTGER4PTGER2L3MBTL1POLBMEN1
SCHEMBL6169204 0.81 ACACB (0.43) POLBCA1CA2ABCB1
SCHEMBL6697114 0.73 HDAC11 (0.43) PTGER4PTGER2POLBCHRM1
SCHEMBL6168074 0.72 RHEB (0.39) PTGER4PTGER2POLBMEN1KMT2A
SCHEMBL6168750 0.71 LMNA (0.46) MEN1KMT2ACA1CA2
SCHEMBL7979501 0.71 L3MBTL1 (0.53) L3MBTL1POLBMEN1KMT2ACA1
SCHEMBL15921100 0.70 KDM4E (0.46) L3MBTL1POLBCCR3
SCHEMBL2062470 0.70 ALDH1A1 (0.59) KMT2A
SCHEMBL6169640 0.70 AR (0.42) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530472-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004014379-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed