SCHEMBL6169640

SCHEMBL6169640

N#Cc1ccc(CN2CC(=O)c3ccc(C(=O)O)cc3C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.42
TSHR P16473 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
COMT P21964 1/20 0.42
CYP2D6 P10635 6/20 0.41
CYP3A4 P08684 6/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
ACHE P22303 1/20 0.41
FAAH O00519 1/20 0.41
USP2 O75604 5/20 0.41
CYP2C19 P33261 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6168895 0.87 CYP3A4 (0.47) TSHRCYP1A2CYP2C9MEN1KMT2A
SCHEMBL6765858 0.82 MEN1 (0.46) ARMEN1KMT2AHDAC1HDAC8
SCHEMBL6168750 0.81 LMNA (0.46) MEN1KMT2APRMT5WDR77
SCHEMBL6167006 0.80 ALDH1A1 (0.42) TSHRCYP2C9MEN1KMT2ACYP2D6
SCHEMBL13630836 0.80 LTA4H (0.56) MEN1KMT2ACYP2D6CYP3A4SMN1; SMN2
Hydrochloric Acid SCHEMBL1075307 0.79 LTA4H (0.55) MEN1KMT2ACYP2D6CYP3A4SMN1; SMN2
SCHEMBL6168074 0.79 RHEB (0.39) MEN1KMT2AACHE
SCHEMBL6167129 0.77 XDH (0.43)
SCHEMBL5012362 0.74 KMT2A (0.71) MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL2722964 0.73 MEN1 (0.49) MEN1KMT2ASMN1; SMN2ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530472-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004014379-A1 ISOQUINOLINE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed