SCHEMBL6173243

SCHEMBL6173243

CC(c1ccncc1NS(=O)(=O)Cc1ccccc1)C1NC(=O)N(c2ccc(S(=O)(=O)C(F)(F)F)cc2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.37
IGF1R P08069 2/20 0.36
ELANE P08246 2/20 0.35
LMNA P02545 1/20 0.35
NAMPT P43490 2/20 0.33
PTGS1 P23219 4/20 0.33
PTGS2 P35354 3/20 0.33
RXFP1 Q9HBX9 1/20 0.32
F2 P00734 1/20 0.31
GLO1 Q04760 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174151 0.90 NAMPT (0.35) IGF1RELANELMNANAMPTPTGS1
SCHEMBL6173841 0.88 LIPE (0.41) METAP2ELANELMNA
SCHEMBL6176687 0.87 IGF1R (0.33) IGF1RLMNA
SCHEMBL6174116 0.87 IGF1R (0.33) IGF1RLMNAPTGS1PTGS2
SCHEMBL6174557 0.86 IGF1R (0.33) IGF1RLMNAPTGS1PTGS2
SCHEMBL6171910 0.85 NAMPT (0.47) ELANENAMPT
SCHEMBL6176021 0.85 IGF1R (0.34) IGF1RLMNAPTGS1PTGS2RXFP1
SCHEMBL6175990 0.83 KIF11 (0.37) IGF1RLMNANAMPTRXFP1
SCHEMBL6174450 0.83 IGF1R (0.38) IGF1RLMNANAMPTRXFP1
SCHEMBL6174089 0.83 GAA (0.36) IGF1RLMNANAMPTRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1599464-A2 NOVEL CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-11-30 EP disclosed
WO-2004070050-A2 CYCLIC UREA DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL USE OF SAME AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-08-19 WO disclosed