SCHEMBL6179366

SCHEMBL6179366

CCc1cc(C(Br)C=O)ccc1F

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SHBG P04278 1/20 0.36
DPP4 P27487 1/20 0.33
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
SLC9A1 P19634 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180857 0.86 SHBG (0.39) SHBG
SCHEMBL27605507 0.81 SHBG (0.33) SHBGDPP4CHRM2CHRM1CHRM3
SCHEMBL27624604 0.80 DPP4 (0.32) SHBGDPP4
SCHEMBL998053 0.80 CES2 (0.42) SHBG
SCHEMBL8772654 0.79 ESR1 (0.43) SHBG
SCHEMBL15017386 0.79 AKR1C3 (0.35) SHBG
SCHEMBL6865041 0.77 VCP (0.38)
SCHEMBL13185576 0.76 TRPV4 (0.35) SHBGDPP4SLC9A1
SCHEMBL18929486 0.76 HSP90AA1 (0.38) SHBGDPP4
SCHEMBL1701138 0.75 MDM2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507530-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2005-02-23 EP disclosed
WO-2003097048-A1 DIAMINOTHIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2003-11-27 WO disclosed