SCHEMBL6184029

SCHEMBL6184029

NC(=O)Nc1ccc(Br)cc1-c1nnn[nH]1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
GPR35 Q9HC97 17/20 0.40
KIF11 P52732 1/20 0.36
KCNMA1 Q12791 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6258779 0.84 CSF1R (0.34)
SCHEMBL27721400 0.84 NPC1 (0.41) GPR35
SCHEMBL1463379 0.84 CXCR1 (0.49) HIF1ANPSR1RXFP1GPR35
SCHEMBL1463507 0.83 KMT2A (0.45)
SCHEMBL1462965 0.82 DDX3X (0.44) HIF1ANPSR1RXFP1GPR35
SCHEMBL1462410 0.82 RAB9A (0.51) GPR35
SCHEMBL1464054 0.82 KMT2A (0.51) GPR35
SCHEMBL6231660 0.81 ALDH1A1 (0.41) GPR35
SCHEMBL27416023 0.81 HIF1A (0.40) HIF1ANPSR1RXFP1GPR35
SCHEMBL27449399 0.81 KIF11 (0.46) GPR35KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101287456-A Diphenylurea derivatives useful as potassium channel activators NEUROSEARCH AS (DK) 2008-10-15 CN claimed
JP-2005538152-A 2005-12-15 JP claimed
EP-1537075-A2 DIARYLUREA DERIVATIVES AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 2005-06-08 EP claimed
WO-2004022529-A2 DIARYLUREA DERIVATIVES AND THEIR USE AS CHLORIDE CHANNEL BLOCKERS NEUROSEARCH A/S (DK) 2004-03-18 WO claimed
EP-1123274-A1 SUBSTITUTED PHENYL DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 2001-08-16 EP claimed
WO-2000024707-A1 SUBSTITUTED PHENYL DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 2000-05-04 WO claimed
CN-101287456-A Diphenylurea derivatives useful as potassium channel activators NEUROSEARCH AS (DK) 2008-10-15 CN disclosed
WO-2004012733-A9 COMPOUNDS USEFUL FOR THE TREATMENT OF DISEASES RESPONSIVE TO ANTIANGIOGENETIC THERAPY NEUROSEARCH AS (DK) 2005-03-10 WO disclosed
WO-2002039987-A2 USE OF MALARIA PARASITE ANION CHANNEL BLOCKERS FOR TREATING MALARIA NEUROSEARCH A/S (DK) 2002-05-23 WO disclosed