SCHEMBL6196196

SCHEMBL6196196

CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)N1CCO[C@](CCOS(C)(=O)=O)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.39
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
WNT3 P56703 2/20 0.37
SFRP1 Q8N474 2/20 0.37
OPRK1 P41145 1/20 0.37
UCHL1 P09936 2/20 0.36
CCR5 P51681 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6196190 0.90 ALDH1A1 (0.42) ALDH1A1HSD17B10HRH2HRH1MEN1
SCHEMBL6198501 0.89 ALDH1A1 (0.43) ALDH1A1HSD17B10HRH2HRH1MEN1
SCHEMBL6197643 0.87 RECQL (0.43) CCR5
SCHEMBL6196499 0.83 CCR5 (0.39) MEN1TSHRKMT2ACCR5
SCHEMBL6202591 0.83 TACR2 (0.38) MEN1TSHRKMT2ACCR5
SCHEMBL6199169 0.83 TACR2 (0.39) MEN1TSHRKMT2ACCR5
SCHEMBL6201334 0.82 CCR5 (0.39) MEN1TSHRKMT2ACCR5
SCHEMBL8113330 0.80 TACR2 (0.35) MEN1TSHRKMT2A
SCHEMBL6197638 0.77 RECQL (0.43) CCR5
SCHEMBL4630697 0.77 TACR2 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1048658-B1 ALICYCLIC ACYLATED HETEROCYCLIC DERIVATIVES SANKYO CO (JP) 2005-06-15 EP disclosed
US-6288059-B1 ANTIASTHMATIC, ANTIALLERGEN AGENTS; URINARY INCONTINENCE; NATURAL KILLER CELL RECEPTOR AND TACHYKININ ANTAGONISTS SANKYO COMPANY, LIMITED (JP) 2001-09-11 US disclosed