SCHEMBL6198119

SCHEMBL6198119

COC(=O)C1=C(CBr)N(C(=O)Oc2ccc([N+](=O)[O-])cc2)C(=O)NC1c1ccc(F)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.38
ADRA1A P35348 2/20 0.38
ADRA1B P35368 2/20 0.38
ADORA3 P0DMS8 1/20 0.37
KDM1A O60341 1/20 0.36
MGLL Q99685 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.35
SLC6A3 Q01959 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577372 0.92 ADORA3 (0.41) ADRA1DADRA1AADRA1BADORA3KDM1A
SCHEMBL7747394 0.92 ADORA3 (0.41) ADRA1DADRA1AADRA1BADORA3KDM1A
SCHEMBL6196041 0.88 ALDH1A1 (0.41) ADRA1DADRA1AADRA1BADORA3MGLL
SCHEMBL6198625 0.78 ADRA1D (0.45) ADRA1DADRA1AADRA1B
SCHEMBL7162576 0.74 ADRA1D (0.54) ADRA1DADRA1AADRA1B
SCHEMBL6193641 0.74 ADRA1D (0.54) ADRA1DADRA1AADRA1B
SCHEMBL7991592 0.73 ADRA1D (0.43) ADRA1DADRA1AADRA1BADORA3MAPT
SCHEMBL6196834 0.73 ADRA1D (0.51) ADRA1DADRA1AADRA1B
SCHEMBL7674379 0.73 ADRA1D (0.51) ADRA1DADRA1AADRA1B
SCHEMBL6956458 0.71 MGLL (0.40) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021185-A4 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMA CORP (US) 2005-09-07 EP disclosed
EP-1021185-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 2000-07-26 EP disclosed
EP-0790826-A4 DIHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMA CORP (US) 1998-11-11 EP disclosed
WO-1997042956-A1 DIDHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-11-20 WO disclosed
EP-0790826-A1 DIHYDROPYRIMIDINES AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1997-08-27 EP disclosed